Brief Information of the Compound and Protein
Compound Name
ethyl 2-[(4R)-4-[[2-benzyl-3-(hydroxyamino)-3-oxopropanoyl]amino]-3-oxo-4,5-dihydro-1H-2-benzazepin-2-yl]acetate
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PubChem ID
CID: 137634777
Canonical SMILES
CCOC(=O)CN1Cc2ccccc2C[C@@H](NC(=O)C(Cc2ccccc2)C(=O)NO)C1=O
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Compound Formula C24H27N3O6
Compound Structure
Protein Name
Histamine H4 receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Histamine receptor
Uniprot ID
Q9H3N8
Gene Name
HRH4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 3018 nM
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