Brief Information of the Compound and Protein
Compound Name
 Compound Info 
US9416103, TV-5-157
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 PubChem ID
CID: 71683085
Canonical SMILES
CCCCn1cc(C(=O)c2cccc3ccccc23)c2cccc(OC)c12
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Compound Formula C24H23NO2
Compound Structure
Protein Name
 Protein Info 
Cannabinoid receptor 1
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Lipid-like ligand receptor (family A GPCR)
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Cannabinoid receptor
Uniprot ID
P47746
Gene Name
CNR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  2
1
IC50 = 45 nM
   TI
   LI
   LO
   TS
2
Ki = 1.7 nM
   TI
   LI
   LO
   TS
CL000020 Neuro-2a
 Cell Line Info 
Mus musculus (Mouse)  2
1
IC50 = 45 nM
   TI
   LI
   LO
   TS
2
Ki = 1.7 nM
   TI
   LI
   LO
   TS