Brief Information of the Compound and Protein
Compound Name
 Compound Info 
5-[[2,6-difluoro-4-(2-methylindazol-5-yl)phenyl]methyl]-6,7-dihydropyrazolo[1,5-a]pyrazin-4-one
    Show/Hide
 PubChem ID
CID: 127050528
Canonical SMILES
Cn1cc2cc(ccc2n1)-c1cc(F)c(CN2CCn3nccc3C2=O)c(F)c1
    Show/Hide
Compound Formula C21H17F2N5O
Compound Structure
Protein Name
 Protein Info 
Muscarinic acetylcholine receptor M1
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Small molecule receptor (family A GPCR)
>
Monoamine receptor
>
Acetylcholine receptor
Uniprot ID
P08482
Gene Name
CHRM1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
EC50 = 1700 nM
   TI
   LI
   LO
   TS