Brief Information of the Compound and Protein
Compound Name
Prx-03140
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PubChem ID
CID: 54677674
SID: 16735420
Canonical SMILES
CC(C)n1c2sccc2c(O)c(C(=O)NCCCN2CCCCC2)c1=O
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Compound Formula C19H27N3O3S
Compound Structure
Protein Name
5-hydroxytryptamine receptor 4
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Serotonin receptor
Uniprot ID
Q13639
Gene Name
HTR4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
EC50 = 58 nM
   TI
   LI
   LO
   TS
CL000053 COS-7 Chlorocebus aethiops (Green monkey)  1
1
EC50 = 17 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 EC50 = 17 nM