Brief Information of the Compound and Protein
Compound Name
2-[3-fluoro-4-[[(1R,2R)-2-[1-[5-(methoxymethyl)pyrimidin-2-yl]piperidin-4-yl]cyclopropyl]methoxymethyl]phenyl]-1-morpholin-4-ylethanone
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PubChem ID
CID: 90116115
Canonical SMILES
COCc1cnc(nc1)N1CCC(CC1)[C@H]1C[C@H]1COCc1ccc(CC(=O)N2CCOCC2)cc1F
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Compound Formula C28H37FN4O4
Compound Structure
Protein Name
Glucose-dependent insulinotropic receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Lipid-like ligand receptor (family A GPCR)
Uniprot ID
Q8TDV5
Gene Name
GPR119
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
EC50 = 3.2 nM
   TI
   LI
   LO
   TS