Brief Information of the Compound and Protein
Compound Name
 Compound Info 
(3R)-5-fluoro-3-hydroxy-3-[[4-(1,2,3,4-tetrahydropyrido[2,3-b]pyrazin-6-ylmethylamino)-2-oxabicyclo[2.2.2]octan-1-yl]methyl]-1,7-diazatricyclo[6.3.1.04,12]dodeca-4(12),5,7,9-tetraen-11-one
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 PubChem ID
CID: 118736762
Canonical SMILES
O[C@@]1(CC23CCC(CC2)(CO3)NCc2ccc3NCCNc3n2)Cn2c3c1c(F)cnc3ccc2=O
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Compound Formula C26H29FN6O3
Compound Structure
Protein Name
 Protein Info 
Potassium voltage-gated channel subfamily H member 2
Protein Classification
Ion channel
>
Voltage-gated ion channel
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Potassium channels
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Voltage-gated potassium channel
Uniprot ID
Q12809
Gene Name
KCNH2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
IC50 > 60000 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 > 60000 nM