Brief Information of the Compound and Protein
Compound Name
[2H]-(S)-methyl 8-(3-fluorobenzyl)-2-(hydroxymethyl)-3-(4-(trifluoromethyl)phenyl)-7,8-dihydro-6H-pyrazolo[1,5-a]pyrrolo[3,4-e]pyrimidine-8-carboxylate
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PubChem ID
CID: 118720428
Canonical SMILES
[2H]C([2H])(O)c1nn2c3c(cnc2c1-c1ccc(C(F)(F)F)cc1)CN[C@]3(Cc1cccc(F)c1)C(=O)OC
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Compound Formula C25H20F4N4O3
Compound Structure
Protein Name
Glucose-dependent insulinotropic receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Lipid-like ligand receptor (family A GPCR)
Uniprot ID
Q8TDV5
Gene Name
GPR119
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
EC50 = 2 nM
   TI
   LI
   LO
   TS