Brief Information of the Compound and Protein
Compound Name
 Compound Info 
5-[4-(1-cyclobutylpiperidin-4-yl)oxyphenyl]-3-ethyl-3,4-diazabicyclo[4.1.0]hept-4-en-2-one
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 PubChem ID
CID: 59652059
Canonical SMILES
CCN1N=C(C2CC2C1=O)c1ccc(OC2CCN(CC2)C2CCC2)cc1
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Compound Formula C22H29N3O2
Compound Structure
Protein Name
 Protein Info 
Histamine H3 receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Histamine receptor
Uniprot ID
Q9Y5N1
Gene Name
HRH3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
Ki = 4.5 nM
   TI
   LI
   LO
   TS