Brief Information of the Compound and Protein
Compound Name
4-[3-[6-(2-methoxyethyl)pyridin-3-yl]-2-methylimidazo[1,2-b]pyridazin-8-yl]morpholine
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PubChem ID
CID: 51352628
SID: 121271484
Canonical SMILES
COCCc1ccc(cn1)-c1c(C)nc2c(ccnn12)N1CCOCC1
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Compound Formula C19H23N5O2
Compound Structure
Protein Name
cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A
Protein Classification
Enzyme
>
Phosphodiesterase
>
Phosphodiesterase 10
>
Phosphodiesterase 10A
Uniprot ID
Q9QYJ6
Gene Name
PDE10A
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000012 Sf21 Spodoptera frugiperda (Fall armyworm)  1
1
IC50 = 58 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 Ki ~ 19 nM