Brief Information of the Compound and Protein
Compound Name
 Compound Info 
N-[(3S)-5,6-dichloro-3-(4-chlorophenyl)-2-oxo-1H-indol-3-yl]-2-(4-methylpiperazin-1-yl)acetamide
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 PubChem ID
CID: 71453404
Canonical SMILES
CN1CCN(CC(=O)N[C@@]2(C(=O)Nc3cc(Cl)c(Cl)cc23)c2ccc(Cl)cc2)CC1
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Compound Formula C21H21Cl3N4O2
Compound Structure
Protein Name
 Protein Info 
Growth hormone secretagogue receptor type 1
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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GRP-related receptor
Uniprot ID
Q92847
Gene Name
GHSR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000643 CHO-K1/CRE-Luc
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  2
1
IC50 = 47 nM
   TI
   LI
   LO
   TS
2
Ki = 249 nM
   TI
   LI
   LO
   TS