Brief Information of the Compound and Protein
Compound Name
N-(4-fluorophenyl)-1-[4-(trifluoromethyl)phenyl]-3,4-dihydro-1H-pyrrolo[1,2-a]pyrazine-2-carboxamide
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PubChem ID
CID: 57326016
SID: 136327987
Canonical SMILES
Fc1ccc(NC(=O)N2CCn3cccc3C2c2ccc(cc2)C(F)(F)F)cc1
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Compound Formula C21H17F4N3O
Compound Structure
Protein Name
Transient receptor potential cation channel subfamily M member 8
Protein Classification
Ion channel
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Voltage-gated ion channel
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Transient receptor potential channel
Uniprot ID
Q8R455
Gene Name
TRPM8
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 180 nM
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