Brief Information of the Compound and Protein
Compound Name
1-[[4-[4-[(1S)-4-(4-methoxyphenoxy)-1-[(2S)-2-methylpyrrolidin-1-yl]butyl]phenyl]phenyl]methyl]piperidine
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PubChem ID
CID: 57328213
SID: 136330355
Canonical SMILES
COc1ccc(OCCC[C@H](N2CCC[C@@H]2C)c2ccc(cc2)-c2ccc(CN3CCCCC3)cc2)cc1
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Compound Formula C34H44N2O2
Compound Structure
Protein Name
Histamine H3 receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Histamine receptor
Uniprot ID
Q9Y5N1
Gene Name
HRH3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000074 SK-N-MC Homo sapiens (Human)  1
1
Ki = 2.042 nM
   TI
   LI
   LO
   TS