Brief Information of the Compound and Protein
Compound Name
4-[4-(4-chlorophenyl)piperidin-1-yl]-1-(3-methylsulfonyl-1,2,4,5-tetrahydro-3-benzazepin-7-yl)butan-1-one
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PubChem ID
CID: 57401509
Canonical SMILES
CS(=O)(=O)N1CCc2ccc(cc2CC1)C(=O)CCCN1CCC(CC1)c1ccc(Cl)cc1
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Compound Formula C26H33ClN2O3S
Compound Structure
Protein Name
Melanin-concentrating hormone receptor 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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MCH receptor
Uniprot ID
P97639
Gene Name
MCHR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 8.5 nM
   TI
   LI
   LO
   TS