Brief Information of the Compound and Protein
Compound Name
2-methyl-4-[4-(3-piperidin-1-ylpropoxy)phenyl]-5,6,7,8-tetrahydrophthalazin-1-one
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PubChem ID
CID: 56658548
Canonical SMILES
Cn1nc(-c2ccc(OCCCN3CCCCC3)cc2)c2CCCCc2c1=O
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Compound Formula C23H31N3O2
Compound Structure
Protein Name
Histamine H3 receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Histamine receptor
Uniprot ID
Q9Y5N1
Gene Name
HRH3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 1.5 nM
   TI
   LI
   LO
   TS