Brief Information of the Compound and Protein
Compound Name
 Compound Info 
1-[(1-cyclopropyl-2-methylpropyl)amino]-7-(1-methylpyrazol-4-yl)-5H-pyrido[4,3-b]indole-4-carboxamide
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 PubChem ID
CID: 42635982
SID: 81075027
Canonical SMILES
CC(C)C(Nc1ncc(C(N)=O)c2[nH]c3cc(ccc3c12)-c1cnn(C)c1)C1CC1
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Compound Formula C23H26N6O
Compound Structure
Protein Name
 Protein Info 
Tyrosine-protein kinase JAK2
Protein Classification
Enzyme
>
Kinase
>
Protein Kinase
>
TK protein kinase group
>
Tyrosine protein kinase JakB family
Uniprot ID
O60674
Gene Name
JAK2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000082 HEL
 Cell Line Info 
Homo sapiens (Human)  1
1
IC50 = 95 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 3 nM