Brief Information of the Compound and Protein
Compound Name
5-[7-Chloro-3-(3,5-dimethylphenyl)-4-{2-[(2R)-piperidin-2-yl]ethoxy}quinolin-6-yl]pyridin-2(1H)-one
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PubChem ID
CID: 52936721
SID: 123076642
Canonical SMILES
Cc1cc(C)cc(c1)-c1cnc2cc(Cl)c(cc2c1OCC[C@H]1CCCCN1)-c1ccc(=O)[nH]c1
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Compound Formula C29H30ClN3O2
Compound Structure
Protein Name
Somatostatin receptor type 2
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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Somatostatin receptor
Uniprot ID
P30874
Gene Name
SSTR2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
IC50 = 0.29 nM
   TI
   LI
   LO
   TS
2
Ki = 0.27 nM
   TI
   LI
   LO
   TS