Brief Information of the Compound and Protein
Compound Name
[3-[7-chloro-6-(1-methylpyrazol-4-yl)-4-[2-[(2R)-piperidin-2-yl]ethoxy]quinolin-3-yl]phenyl]methanol
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PubChem ID
CID: 52936830
SID: 123076758
Canonical SMILES
Cn1cc(cn1)-c1cc2c(OCC[C@H]3CCCCN3)c(cnc2cc1Cl)-c1cccc(CO)c1
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Compound Formula C27H29ClN4O2
Compound Structure
Protein Name
Somatostatin receptor type 2
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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Somatostatin receptor
Uniprot ID
P30874
Gene Name
SSTR2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
IC50 = 8.3 nM
   TI
   LI
   LO
   TS
2
Ki = 0.13 nM
   TI
   LI
   LO
   TS