Brief Information of the Compound and Protein
Compound Name
(S)-7-chloro-3-(3,5-dimethylphenyl)-6-(1-methyl-1H-pyrazol-4-yl)-4-(2-(piperidin-2-yl)ethoxy)quinoline
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PubChem ID
CID: 24951595
SID: 56249395
Canonical SMILES
Cc1cc(C)cc(c1)-c1cnc2cc(Cl)c(cc2c1OCC[C@@H]1CCCCN1)-c1cnn(C)c1
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Compound Formula C28H31ClN4O
Compound Structure
Protein Name
Somatostatin receptor type 2
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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Somatostatin receptor
Uniprot ID
P30874
Gene Name
SSTR2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
IC50 = 145 nM
   TI
   LI
   LO
   TS
2
Ki = 1.5 nM
   TI
   LI
   LO
   TS