Brief Information of the Compound and Protein
Compound Name
5-methyl-2-[(5-methyl-1H-imidazol-4-yl)methyl]-3,4-dihydropyrid[4,3-b]indol-1-one;hydrochloride
    Show/Hide
PubChem ID
CID: 2099
SID: 14922649
Canonical SMILES
Cc1nc[nH]c1CN1CCc2c(C1=O)c1ccccc1n2C
    Show/Hide
Compound Formula C17H18N4O
Compound Structure
Protein Name
Potassium voltage-gated channel subfamily H member 2
Protein Classification
Ion channel
>
Voltage-gated ion channel
>
Potassium channels
>
Voltage-gated potassium channel
Uniprot ID
Q12809
Gene Name
KCNH2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 3235.94 nM
   TI
   LI
   LO
   TS
CL000006 HEK293 Homo sapiens (Human)  1
1
IC50 = 2300 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 IC50 = 3200 nM
2 IC50 = 3235.94 nM