Brief Information of the Compound and Protein
Compound Name
(2S,4R,5R)-1,2,5-trimethyl-4-(naphthalen-1-ylethynyl)piperidin-4-ol
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PubChem ID
CID: 52941061
Canonical SMILES
C[C@H]1C[C@](O)(C#Cc2cccc3ccccc23)[C@H](C)CN1C
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Compound Formula C20H23NO
Compound Structure
Protein Name
Histamine H3 receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Histamine receptor
Uniprot ID
Q9Y5N1
Gene Name
HRH3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000156 HT-1080 Homo sapiens (Human)  1
1
IC50 = 41 nM
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