Brief Information of the Compound and Protein
Compound Name
1-(2-hydroxy-5-(1H-tetrazol-5-yl)phenyl)-3-(4-(quinolin-2-ylmethoxy)phenyl)prop-2-en-1-one
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PubChem ID
CID: 135430849
SID: 14881933
Canonical SMILES
O=C(/C=C/c1ccc(OCc2ccc3ccccc3n2)cc1)c1cc(-c2nn[nH]n2)ccc1O
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Compound Formula C26H19N5O3
Compound Structure
Protein Name
Cysteinyl leukotriene receptor 1
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Lipid-like ligand receptor (family A GPCR)
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Leukotriene receptor
Uniprot ID
Q9Y271
Gene Name
CYSLTR1
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000100 U-937 Homo sapiens (Human)  1
1
IC50 = 14 nM
   TI
   LI
   LO
   TS