Brief Information of the Compound and Protein
Compound Name
N-cyclohexyl-4-(1H-imidazol-5-yl)piperidine-1-carbothioamide
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PubChem ID
CID: 3035905
SID: 14922586
Canonical SMILES
S=C(NC1CCCCC1)N1CCC(CC1)c1cnc[nH]1
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Compound Formula C15H24N4S
Compound Structure
Protein Name
Histamine H3 receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Histamine receptor
Uniprot ID
Q9QYN8
Gene Name
HRH3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000049 C6 Rattus norvegicus (Rat)  1
1
Ki = 3.631 nM
   TI
   LI
   LO
   TS
CL000026 CHO-K1 Cricetulus griseus (Chinese hamster)  1
1
Ki = 6.5 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 Ki = 2.65 nM
2 Ki = 3.981 nM
3 Ki = 4 nM