Brief Information of the Compound and Protein
Compound Name
 Compound Info 
(Z)-2-(3-(3-fluoro-4-((4-fluorobenzyl)(pyridin-2-ylmethyl)amino)piperidin-1-yl)-3-oxoprop-1-enyl)benzonitrile
    Show/Hide
 PubChem ID
CID: 46865537
SID: 99304498
Canonical SMILES
N#Cc1ccccc1/C=C\C(=O)N1CCC(N(Cc2ccc(F)cc2)Cc2ccccn2)C(F)C1
    Show/Hide
Compound Formula C28H26F2N4O
Compound Structure
Protein Name
 Protein Info 
Proteinase-activated receptor 1
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Peptide receptor (family A GPCR)
>
Protease-activated receptor
>
Protease-activated receptor
Uniprot ID
P25116
Gene Name
F2R
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
Kd = 588.84 nM
   TI
   LI
   LO
   TS