Brief Information of the Compound and Protein
Compound Name
N-[[3,5-bis(trifluoromethyl)phenyl]methyl]-2-(1-methylsulfonylpiperidin-3-yl)-4-spiro[indene-1,4'-piperidine]-1'-ylbutanamide
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PubChem ID
CID: 44416156
Canonical SMILES
CS(=O)(=O)N1CCCC(C1)C(CCN1CCC2(CC1)C=Cc1ccccc21)C(=O)NCc1cc(cc(c1)C(F)(F)F)C(F)(F)F
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Compound Formula C32H37F6N3O3S
Compound Structure
Protein Name
C-C chemokine receptor type 2
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Chemokine receptor
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CC chemokine receptor
Uniprot ID
P41597
Gene Name
CCR2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
IC50 = 783 nM
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