Brief Information of the Compound and Protein
| Compound Name |
(risperidone)3-{2-[4-(6-Fluoro-benzo[d]isoxazol-3-yl)-piperidin-1-yl]-ethyl}-2-methyl-6,7,8,9-tetrahydro-pyrido[1,2-a]pyrimidin-4-one
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PubChem ID | |||||
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Compound Structure |
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| Protein Name |
D(3) dopamine receptor
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Protein Classification |
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Dopamine receptor
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| Uniprot ID | Gene Name | DRD3 |
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Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Biochemical Assays
| 1 | Ki = 6.7 nM | ||
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| 2 | Ki = 9.6 nM | ||
| 3 | Ki = 13 nM | ||
| 4 | Ki = 14 nM | ||
| 5 | Ki = 14.3 nM | ||
| 6 | Ki = 16 nM | ||
| 7 | Ki = 16.22 nM | ||
| 8 | Ki = 100 nM | ||