Brief Information of the Compound and Protein
Compound Name
1-(4-(3-(piperidin-1-yl)propoxy)phenyl)-4-(pyrazolo[1,5-a]pyrimidine-3-carbonyl)piperazin-2-one formic acid
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PubChem ID
CID: 24748892
SID: 49651012
Canonical SMILES
O=C(c1cnn2cccnc12)N1CCN(c2ccc(OCCCN3CCCCC3)cc2)C(=O)C1.O=CO
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Compound Formula C26H32N6O5
Compound Structure
Protein Name
Histamine H3 receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Histamine receptor
Uniprot ID
Q9Y5N1
Gene Name
HRH3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  1
1
Ki = 3.981 nM
   TI
   LI
   LO
   TS