Brief Information of the Compound and Protein
Compound Name
 Compound Info 
4-(4-(azetidine-1-carbonyl)benzoyl)-1-(4-(1-cyclobutylpiperidin-4-yloxy)phenyl)piperazin-2-one formic acid
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 PubChem ID
CID: 24749292
SID: 49651412
Canonical SMILES
O=C(c1ccc(C(=O)N2CCN(c3ccc(OC4CCN(C5CCC5)CC4)cc3)C(=O)C2)cc1)N1CCC1.O=CO
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Compound Formula C31H38N4O6
Compound Structure
Protein Name
 Protein Info 
Histamine H3 receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Histamine receptor
Uniprot ID
Q9Y5N1
Gene Name
HRH3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  1
1
Ki = 0.3162 nM
   TI
   LI
   LO
   TS