Brief Information of the Compound and Protein
Compound Name
2-amino-N-((S)-2-(benzyloxy)-1-(2-((1-(methylsulfonyl)indolin-2-yl)methyl)-2H-tetrazol-5-yl)ethyl)-2-methylpropanamide
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PubChem ID
CID: 44434078
Canonical SMILES
CC(C)(N)C(=O)N[C@H](COCc1ccccc1)c1nnn(CC2Cc3ccccc3N2S(C)(=O)=O)n1
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Compound Formula C24H31N7O4S
Compound Structure
Protein Name
Growth hormone secretagogue receptor type 1
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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GRP-related receptor
Uniprot ID
Q92847
Gene Name
GHSR
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000008 H4 Homo sapiens (Human)  1
1
EC50 = 546 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 Ki > 5000 nM