Brief Information of the Compound and Protein
Compound Name
(5-(1-isopropylpiperidin-4-yloxy)-2-methyl-1H-indol-3-yl)(morpholino)methanone
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PubChem ID
CID: 44185183
SID: 85180513
Canonical SMILES
CC(C)N1CCC(CC1)Oc1ccc2[nH]c(C)c(C(=O)N3CCOCC3)c2c1
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Compound Formula C22H31N3O3
Compound Structure
Protein Name
Histamine H3 receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Small molecule receptor (family A GPCR)
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Monoamine receptor
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Histamine receptor
Uniprot ID
Q9Y5N1
Gene Name
HRH3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO Cricetulus griseus (Chinese hamster)  2
1
EC50 = 405 nM
   TI
   LI
   LO
   TS
2
Ki = 86 nM
   TI
   LI
   LO
   TS