Brief Information of the Compound and Protein
Compound Name
 Compound Info 
3-((4-(4-chlorophenyl)piperazin-1-yl)methyl)H-pyrazolo[1,5-a]pyridine
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 PubChem ID
CID: 10404144
SID: 15421269
Canonical SMILES
Clc1ccc(cc1)N1CCN(Cc2cnn3ccccc23)CC1
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Compound Formula C18H19ClN4
Compound Structure
Protein Name
 Protein Info 
D(4) dopamine receptor
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Small molecule receptor (family A GPCR)
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Monoamine receptor
>
Dopamine receptor
Uniprot ID
P21917
Gene Name
DRD4
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000011 CHO
 Cell Line Info 
Cricetulus griseus (Chinese hamster)  4
1
EC50 = 12 nM
   TI
   LI
   LO
   TS
2
Ki = 2.291 nM
   TI
   LI
   LO
   TS
3
Ki = 3.1 nM
   TI
   LI
   LO
   TS
4
Ki = 3.6 nM
   TI
   LI
   LO
   TS
Biochemical Assays
1 Ki = 2 nM
2 Ki = 3.6 nM