Brief Information of the Compound and Protein
Compound Name
 Compound Info 
(S)-6-Amino-2-((R)-3-(1H-indol-3-yl)-2-{[4-(2-oxo-2,3-dihydro-benzoimidazol-1-yl)-piperidine-1-carbonyl]-amino}-propionylamino)-hexanoic acid tert-butyl ester
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 PubChem ID
CID: 44325477
Canonical SMILES
CC(C)(C)OC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc1c[nH]c2ccccc12)NC(=O)N1CCC(CC1)n1c2ccccc2[nH]c1=O
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Compound Formula C34H45N7O5
Compound Structure
Protein Name
 Protein Info 
Somatostatin receptor type 2
Protein Classification
Membrane receptor
>
Family A G protein-coupled receptor
>
Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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Somatostatin receptor
Uniprot ID
P30874
Gene Name
SSTR2
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000029 GH4C1
 Cell Line Info 
Rattus norvegicus (Rat)  1
1
IC50 = 6.5 nM
   TI
   LI
   LO
   TS
CL000020 Neuro-2a
 Cell Line Info 
Mus musculus (Mouse)  1
1
IC50 = 0.26 nM
   TI
   LI
   LO
   TS