Brief Information of the Compound and Protein
Compound Name
5-(5-Dimethylamino-naphthalene-1-sulfonylamino)-3-methyl-isoxazole-4-carboxylic acid ethyl ester
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PubChem ID
CID: 10476286
SID: 15500015
Canonical SMILES
CCOC(=O)c1c(C)noc1NS(=O)(=O)c1cccc2c(cccc12)N(C)C
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Compound Formula C19H21N3O5S
Compound Structure
Protein Name
Endothelin-1 receptor
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Short peptide receptor (family A GPCR)
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Endothelin receptor
Uniprot ID
P26684
Gene Name
EDNRA
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000139 A-10 Rattus norvegicus (Rat)  1
1
IC50 = 31000 nM
   TI
   LI
   LO
   TS