Brief Information of the Compound and Protein
| Compound Name |
9-cis retinoic acid
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PubChem ID | |||||
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Compound Structure |
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| Protein Name |
Retinoic acid receptor gamma
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Protein Classification |
Transcription factor
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Nuclear receptor
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Nuclear hormone receptor subfamily 1
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Nuclear hormone receptor subfamily 1 group B
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Nuclear hormone receptor subfamily 1 group B member 3
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| Uniprot ID | Gene Name | RARG |
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Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
| Cell Line ID | Cell Line Name | Cell Line Organism | |
| CL000044 | CV-1 | Chlorocebus aethiops (Green monkey) | 3 |
| 1 |
AC50 = 3 nM
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TI
LI
LO
TS
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| 2 |
EC50 = 45 nM
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TI
LI
LO
TS
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| 3 |
EC50 = 50 nM
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TI
LI
LO
TS
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Biochemical Assays
| 1 | EC50 = 6 nM | ||
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| 2 | EC50 = 12 nM | ||
| 3 | EC50 = 45 nM | ||
| 4 | IC50 = 17 nM | ||
| 5 | Kd = 0.8 nM | ||
| 6 | Kd = 22 nM | ||
| 7 | Kd = 148 nM | ||
| 8 | Kd = 150 nM | ||
| 9 | Ki = 20 nM | ||