General Information of the Protein
Protein ID
PT06742
Protein Name
Gag polyprotein
Gene Name
GAG
Sequence
REEQVTSEQAKFWLGLGGGRVSPPGPECIEKPATERRIDKGEEMGETTVQRDAKMAPEKMATPKTVGTSCYQCGTATGCNCVTASAPPPPYVGSGLYPSLAGAGEQGQGGDTPRGAEQPRAEPGHAGQAPGPALTDWARIREELASTGPPVVAMPVVIKTEGPAWTPLEPEDTRWLDGKHKRKSSQCLVKSSMSGYIPSCLDKDEQCVVCGDKATGYHYRCITCEGCKSFFRRTIQKNLHPTYSCTYDGCCVIDKITRNQCQLCRFKKCISVGMAMDLVLDDSKRVAKRKLIEENRERRRKEEMIKSLQHRPSPSAEEWELIHVVTEAHRSTNAQGSHWKQRRKFLLEDIGQSPMASMLDGDKVDLEAFSEFTKIITPAITRVVDFAKNLPMFSELPCEDQIILLKGCCMEIMSLRAAVRYDPESETLTLSGEMAVKREQLKNGGLGVVSDAIFDLGKSLSAFNLDDTEVALLQAVLLMSSDRTGLICVDKIEKCQESYLLAFEHYINYRKHNIPHFWSKLLMKVADLRMIGAYHASRFLHMKVECPTELSPQEV
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Organism
Avian erythroblastosis virus (strain ES4)
Protein Classification
Surface antigen
Function
Acts as a thyroid-hormone receptor antagonist. The v-ErbA oncogene cooperates with v-ErbB and other primarily sarcoma-inducing oncogenes in transformation of erythroblasts. It is non transforming by itself and cannot induce self-renewal of erythroblasts. Instead it blocks the residual capacity of the v-ErbB cells to differentiate terminally.
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Uniprot ID
Primary ID:
P03373

Secondarily ID:
Q85511
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Subcellular Location
Virion
Map of Molecular Bioactivity Related to the Protein
Map of Molecular Bioactivity Related to the Protein

Protein
Cell Line
Compound

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Protein
Cell Line ID: CL000209 , HEC-1
Compound ID Compound Name Compound Formula
CP0866774
2-[3-chloro-3-phenylprop-2-enylidene]hydrazinecarboximidamide
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C10H11ClN4
 1
1
IC50 = 900 nM
   TI
   LI
   LO
   TS
CP0870866
1-Chloro-5,7-dimethyl-3,4-dihydronaphthalene-2-carboxaldehyde guanylhydrazone
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C14H17ClN4
 1
1
IC50 = 1200 nM
   TI
   LI
   LO
   TS
CP0911608
2-[(3-chloro-1H-inden-2-yl)methylene]hydrazinecarboximidamide
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C11H11ClN4
 1
1
IC50 = 1300 nM
   TI
   LI
   LO
   TS
CP0677046
2-[(1-chloro-3,4-dihydronaphthalen-2-yl)methylene]hydrazinecarboximidamide
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C12H13ClN4
 1
1
IC50 = 1400 nM
   TI
   LI
   LO
   TS
CP0833861
beta-Chloro-alpha-methylcinnamaldehyde guanylhydrazone
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C11H13ClN4
 1
1
IC50 = 1400 nM
   TI
   LI
   LO
   TS
CP0891605
1-Chloro-3-dihydro-4-methylnaphthalene-2-carboxaldehyde guanylhydrazone
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C13H15ClN4
 1
1
IC50 = 1500 nM
   TI
   LI
   LO
   TS
CP0859243
1-Chloro-6-methoxy-3,4-dihydronaphthalene-2-carboxaldehyde guanylhydrazone
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C13H15ClN4O
 1
1
IC50 = 2000 nM
   TI
   LI
   LO
   TS
CP0859244
1-Methoxy-3,4-dihydronaphthalene-2-carboxaldehyde guanylhydrazone
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C13H16N4O
 1
1
IC50 = 3100 nM
   TI
   LI
   LO
   TS
CP0646102
9-Chloro-6,7-dihydro-5-benzocycloheptene-8-carboxaldehyde guanylhydrazone
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C13H15ClN4
 1
1
IC50 = 3300 nM
   TI
   LI
   LO
   TS
CP0870867
1-Phenoxy-3,4-dihydronaphthalene-2-carboxaldehyde guanylhydrazone
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C18H18N4O
 1
1
IC50 = 3500 nM
   TI
   LI
   LO
   TS
CP0849918
1-Chloro-7-methoxy-3,4-dihydronaphthalene-2-carboxaldehyde guanylhydrazone
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C13H15ClN4O
 1
1
IC50 = 3900 nM
   TI
   LI
   LO
   TS
CP0434732
2-[(E)-naphthalen-2-ylmethylideneamino]guanidine
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C12H13ClN4
 1
1
IC50 = 7500 nM
   TI
   LI
   LO
   TS
CP0904375
N''-[(1E)-1-naphthylmethylene]carbonohydrazonic diamide
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C12H12N4
 1
1
IC50 = 7500 nM
   TI
   LI
   LO
   TS
CP0870868
1-Bromo-3,4-dihydronaphthalene-2-carboxaldehyde guanylhydrazone
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C12H13BrN4
 1
1
IC50 = 7800 nM
   TI
   LI
   LO
   TS
CP0877207
1-(1,1,1,Trifluoromethyl)-3,4-dihydronaphthalene-2-carboxaldehyde guanylhydrazone
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C13H13F3N4
 1
1
IC50 = 12000 nM
   TI
   LI
   LO
   TS
CP0849912
3-Chloro-3-naphthalen-1-yl-propenal guanylhydrazone
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C14H13ClN4
 1
1
IC50 >= 50000 nM
   TI
   LI
   LO
   TS
CP0877205
1-(1-Chloro-3,4-dihydro-naphthalen-2-yl)-ethanone guanylhydrazone
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C13H15ClN4
 1
1
IC50 >= 50000 nM
   TI
   LI
   LO
   TS
Similar Protein(s) and Bioactivity Statistics
50% Identity
Protein ID Protein Name Protein Organism
PT01591 Thyroid hormone receptor alpha Homo sapiens, Human