General Information of the Protein
Protein ID
PT06702
Protein Name
Taste receptor type 2 member 16
Gene Name
TAS2R16
Sequence
MIPIQLTVFFMIIYVLESLTIIVQSSLIVAVLGREWLQVRRLMPVDMILISLGISRFCLQWASMLNNFCSYFNLNYVLCNLTITWEFFNILTFWLNSLLTVFYCIKVSSFTHHIFLWLRWRILRLFPWILLGSLMITCVTIIPSAIGNYIQIQLLTMEHLPRNSTVTDKLENFHQYQFQAHTVALVIPFILFLASTIFLMASLTKQIQHHSTGHCNPSMKARFTALRSLAVLFIVFTSYFLTILITIIGTLFDKRCWLWVWEAFVYAFILMHSTSLMLSSPTLKRILKGKC
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Organism
Homo sapiens, Human
Protein Classification
Membrane receptor
>
Taste family G protein-coupled receptor
>
Taste receptor (taste family GPCR)
Function
Gustducin-coupled receptor implicated in the perception of bitter compounds in the oral cavity and the gastrointestinal tract. Signals through PLCB2 and the calcium-regulated cation channel TRPM5.
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Uniprot ID
Primary ID:
Q9NYV7

Secondarily ID:
A4D0X2
Q502V3
Q549U8
Q645W1
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HGNC ID
HGNC:14921
Subcellular Location
Cell membrane
Map of Molecular Bioactivity Related to the Protein
Map of Molecular Bioactivity Related to the Protein

Protein
Cell Line
Compound

Bioactivity Value:

<= 0.1 μM
> 0.1 μM and <= 10 μM
> 10 μM
Imprecise Activity
Table of Molecular Bioactivities Related to the Protein
Cell Line ID: CL000902 , HEK293/Galpha15
Compound ID Compound Name Compound Formula
CP0194955
CHEBI:17814
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C13H18O7
 1
1
Activity = 70000 nM
   TI
   LI
   LO
   TS
CP0411348
phenyl-beta-d-glucopyranoside
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C12H16O6
 1
1
Activity = 70000 nM
   TI
   LI
   LO
   TS
CP0905710
helicin
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C13H16O7
 1
1
Activity = 300000 nM
   TI
   LI
   LO
   TS
CP0900071
beta-Naphthyl-beta-D-glucopyranoside
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C16H18O6
 1
1
Activity = 400000 nM
   TI
   LI
   LO
   TS
CP0039774
4-hydroxyphenyl beta-D-glucopyranoside
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C12H16O7
 1
1
Activity = 500000 nM
   TI
   LI
   LO
   TS
CP0895836
2-nitro-phenyl-beta-D-glucopyranoside
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C12H15NO8
 1
1
Activity = 1500000 nM
   TI
   LI
   LO
   TS
CP0669553
Amygdalin
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C20H27NO11
 1
1
Activity = 2300000 nM
   TI
   LI
   LO
   TS
CP0040072
CHEBI:4853
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C15H16O9
 1
1
Activity = 4000000 nM
   TI
   LI
   LO
   TS
CP0109401
CHEBI:320055
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C7H14O6
 1
1
Activity = 15000000 nM
   TI
   LI
   LO
   TS