Brief Information of the Cell Line and Protein
Cell Line ID: CL000659 , UMR-106
Synonyms
UMR 106
UMR106
Category Cancer cell line
Organism
Rattus norvegicus (Rat)
Cellosaurus ID
CVCL_3617
Protein ID: PT06582 , Parathyroid hormone/parathyroid hormone-related peptide receptor
Gene Name PTH1R
Organism Rattus norvegicus, Rat
Protein Classification Membrane receptor
Uniprot ID P25961
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000659  Protein ID: PT06582
 
Compound ID Compound Name Compound Formula
CP0398972
Aib-Val-Aib-Glu-lle-Gln-Leu-Nle-His-Gln-Arg-Ala-Lys-Tyr
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C76H127N23O19
 1
1
EC50 = 1.1 nM
   TI
   LI
   LO
   TS
CP0431771
Ala-Val-Ala-Glu-lle-Gln-Leu-Nle-His-Gln-Har-Ala-Lys-Trp-Tyr
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C86H135N25O20
 1
1
EC50 = 129 nM
   TI
   LI
   LO
   TS
CP0436332
Ala-Val-Ala-Glu-lle-Gln-Leu-Met-His-Gln-Har-Ala-Lys-Trp
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C76H124N24O18S
 1
1
EC50 = 155 nM
   TI
   LI
   LO
   TS
CP0423354
Ala-Val-Ala-Glu-lle-Gln-Leu-Met-His-Gln-Har-Ala-Lys-Trp-Fly
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C102H146N26O23S
 1
1
EC50 = 251 nM
   TI
   LI
   LO
   TS
CP0431898
Ala-Val-Ala-Glu-lle-Gln-Leu-Nle-His-Gln-Har-Ala-Lys-Tyr
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C75H125N23O19
 1
1
EC50 = 344 nM
   TI
   LI
   LO
   TS