Brief Information of the Cell Line and Protein
Cell Line ID: CL001015 , CHO CRE-SPAP
Category Spontaneously immortalized cell line
Organism
Cricetulus griseus (Chinese hamster)
Cellosaurus ID
CVCL_0213
Protein ID: PT05120 , Transmembrane domain-containing protein TMIGD3
Gene Name TMIGD3
Organism Homo sapiens, Human
Protein Classification Unclassified protein
Uniprot ID P0DMS9
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL001015  Protein ID: PT05120
 
Compound ID Compound Name Compound Formula
CP0386349
6-ethyl-2-(furan-3-yl)-3H-thieno[2,3-d]pyrimidin-4-one
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C12H10N2O2S
 2
1
Kd = 741.31 nM
   TI
   LI
   LO
   TS
2
Ki = 549.54 nM
   TI
   LI
   LO
   TS
CP0406250
N-(4-cyclopropyl-1,3-thiazol-2-yl)-1-benzothiophene-2-carboxamide
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C15H12N2OS2
 1
1
Kd = 741.31 nM
   TI
   LI
   LO
   TS
CP0567375
2,5-bis(furan-2-yl)-3H-thieno[2,3-d]pyrimidin-4-one
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C14H8N2O3S
 1
1
Ki = 138.04 nM
   TI
   LI
   LO
   TS
CP0472633
N-(1,3-benzothiazol-2-yl)-1-benzothiophene-2-carboxamide
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C16H10N2OS2
 1
1
Ki = 331.13 nM
   TI
   LI
   LO
   TS
CP0429824
MLS-0463381.0001
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C15H12N2OS2
 1
1
Ki = 380.19 nM
   TI
   LI
   LO
   TS
CP0544928
2-(furan-3-yl)-5,6-dimethyl-3H-thieno[2,3-d]pyrimidin-4-one
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C12H10N2O2S
 1
1
Ki = 398.11 nM
   TI
   LI
   LO
   TS
CP0395100
2-cyclopropyl-6-ethyl-3H-thieno[2,3-d]pyrimidin-4-one
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C11H12N2OS
 1
1
Ki = 1819.7 nM
   TI
   LI
   LO
   TS
CP0447828
6-ethyl-2-pyridin-4-yl-3H-thieno[2,3-d]pyrimidin-4-one
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C13H11N3OS
 1
1
Ki = 1995.26 nM
   TI
   LI
   LO
   TS
CP0429823
3-methyl-N-(4-methyl-5-methylsulfanyl-1,3-thiazol-2-yl)but-2-enamide
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C10H14N2OS2
 1
1
Ki = 2187.76 nM
   TI
   LI
   LO
   TS
CP0420582
6-ethyl-2-pyrrolidin-1-yl-3H-thieno[2,3-d]pyrimidin-4-one
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C12H15N3OS
 1
1
Ki = 2290.87 nM
   TI
   LI
   LO
   TS
CP0452183
N-(1H-indazol-5-yl)-1H-pyrrole-2-carboxamide
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C12H10N4O
 1
1
Ki = 2398.83 nM
   TI
   LI
   LO
   TS
CP0540845
N-(4-cyclopropyl-1,3-thiazol-2-yl)-2,2-dimethylpropanamide
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C11H16N2OS
 1
1
Ki = 4897.79 nM
   TI
   LI
   LO
   TS
CP0508748
6-Ethyl-thieno[2,3-d]pyrimidin-4-ol
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C8H8N2OS
 1
1
Ki = 13489.63 nM
   TI
   LI
   LO
   TS