Brief Information of the Cell Line and Protein
Cell Line ID: CL000902 , HEK293/Galpha15
 Cell Line Info 
Category Transformed cell line
Organism
Homo sapiens (Human)
Protein ID: PT04808 , Proteinase-activated receptor 4
 Protein Info 
Gene Name F2RL3
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID Q96RI0
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000902
 Cell Line Info 
 Protein ID: PT04808
 Protein Info 
 
Compound ID Compound Name Compound Formula
CP0551164
 Compound Info 
8-(4-chloro-6-methoxy-1,3-benzothiazol-2-yl)-3,6-dimethylquinazolin-4-one
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C18H14ClN3O2S
  1
1
IC50 = 0.53 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0479453
 Compound Info 
US10047103, 94
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C23H23N5O5S2
  1
1
IC50 = 0.7 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0549763
 Compound Info 
N-[2-[[4-chloro-2-(3,6-dimethyl-4-oxoquinazolin-8-yl)-1,3-benzothiazol-6-yl]oxy]ethyl]-4-(trifluoromethyl)benzenesulfonamide
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C26H20ClF3N4O4S2
  1
1
IC50 = 1.2 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0491440
 Compound Info 
8-(4-fluoro-6-methoxy-1,3-benzothiazol-2-yl)-3,6-dimethylquinazolin-4-one
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C18H14FN3O2S
  1
1
IC50 = 3.2 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0471307
 Compound Info 
3,6-dimethyl-8-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)quinazolin-4-one
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C17H17N3OS
  1
1
IC50 = 5.7 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS
CP0479451
 Compound Info 
8-(4-chloro-6-methoxy-1,3-benzothiazol-2-yl)-6-ethyl-3-methylquinazolin-4-one
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C19H16ClN3O2S
  1
1
IC50 = 6.8 nM
 Bioactivity Info 
   TI
   LI
   LO
   TS