Brief Information of the Compound and Protein
Compound Name
N-[2-[[4-chloro-2-(3,6-dimethyl-4-oxoquinazolin-8-yl)-1,3-benzothiazol-6-yl]oxy]ethyl]-4-(trifluoromethyl)benzenesulfonamide
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Canonical SMILES
Cc1cc(-c2nc3c(Cl)cc(OCCNS(=O)(=O)c4ccc(cc4)C(F)(F)F)cc3s2)c2ncn(C)c(=O)c2c1
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Compound Formula C26H20ClF3N4O4S2
Compound Structure
Protein Name
Proteinase-activated receptor 4
Protein Classification
Membrane receptor
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Family A G protein-coupled receptor
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Peptide receptor (family A GPCR)
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Protease-activated receptor
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Protease-activated receptor
Uniprot ID
Q96RI0
Gene Name
F2RL3
Table of Molecular Bioactivities Related to the Compound and Protein
Cell-based Assay
Cell Line ID Cell Line Name Cell Line Organism
CL000902 HEK293/Galpha15 Homo sapiens (Human)  1
1
IC50 = 1.2 nM
   TI
   LI
   LO
   TS