| Compound ID |
Compound Name |
Compound Formula |
|
CP0495789
|
US11304929, Example 05-017
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|
C24H26Cl2N2O6S
|
1
|
| 1 |
IC50 = 0.3 nM
|
|
|
|
CP0549264
|
US11304929, Example 01-023
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|
C21H21Cl2N3O6S
|
1
|
| 1 |
IC50 = 0.8 nM
|
|
|
|
CP0482900
|
US11304929, Example 05-009
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|
C23H25ClN2O5S
|
1
|
| 1 |
IC50 = 1.6 nM
|
|
|
|
CP0476347
|
ethyl 2-[4-[(1S)-1-[(4,5-dichloro-1,6-dimethylindole-2-carbonyl)amino]-2-hydroxyethyl]phenyl]sulfonylacetate
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|
C23H24Cl2N2O6S
|
1
|
| 1 |
IC50 = 2.9 nM
|
|
|
|
CP0549273
|
US11304929, Example 01-005
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|
C23H25ClN2O6S
|
1
|
| 1 |
IC50 = 3.3 nM
|
|
|
|
CP0429990
|
US11304929, Example 05-010
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|
C26H29ClN2O6S
|
1
|
| 1 |
IC50 = 3.7 nM
|
|
|
|
CP0549265
|
US11304929, Example 05-011
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|
C24H27ClN2O5S
|
1
|
| 1 |
IC50 = 3.9 nM
|
|
|
|
CP0534939
|
US11304929, Example 01-007
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|
C22H22Cl2N2O6S
|
1
|
| 1 |
IC50 = 5 nM
|
|
|
|
CP0551978
|
US11304929, Example 01-001
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|
C22H22Cl2N2O5S
|
1
|
| 1 |
IC50 = 7 nM
|
|
|
|
CP0472976
|
US11304929, Example 01-028
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|
C23H24F2N2O6S
|
1
|
| 1 |
IC50 = 7.3 nM
|
|
|
|
CP0468813
|
US11304929, Example 01-013
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|
C22H23ClN2O6S
|
1
|
| 1 |
IC50 = 8.3 nM
|
|
|
|
CP0540681
|
US11304929, Example 05-004
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|
C25H29ClN2O5S
|
1
|
| 1 |
IC50 = 10.1 nM
|
|
|
|
CP0910388
|
4-chloro-N-[(1R)-1-[4-(3-{4-[(1R)-1-[(4-chloro-1,6-dimethyl-1H-indol-2-yl)formamido]ethyl]benzenesulfonyl}-2-oxopropanesulfonyl)phenyl]ethyl]-1,6-dimethyl-1H-indole-2-carboxamide
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|
C41H40Cl2N4O7S2
|
1
|
| 1 |
IC50 = 11.9 nM
|
|
|
|
CP0540688
|
US11304929, Example 01-021
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|
C24H26Cl2N2O6S
|
1
|
| 1 |
IC50 = 12.6 nM
|
|
|
|
CP0490149
|
US11304929, Example 09-014
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|
C26H29ClN2O6S
|
1
|
| 1 |
IC50 = 14.7 nM
|
|
|
|
CP0558633
|
US11304929, Example 09-011
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|
C29H26ClF3N2O5S
|
1
|
| 1 |
IC50 = 20.1 nM
|
|
|
|
CP0529475
|
(3-methyloxetan-3-yl)methyl 2-{4-[(1R)-1-[(4-chloro-1,6-dimethyl-1H-indol-2- yl)formamido]ethyl]benzenesulfonyl}acetate
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|
C26H29ClN2O6S
|
1
|
| 1 |
IC50 = 22.2 nM
|
|
|
|
CP0531728
|
(acetyloxy)methyl 2-{4-[(1R)-1-[(1-methyl-3-phenyl-1H-pyrazol-5- yl)formamido]ethyl]benzenesulfonyl}acetate
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|
C24H25N3O7S
|
1
|
| 1 |
IC50 = 23.7 nM
|
|
|
|
CP0483823
|
2-hydroxyethyl 2-{4-[(1R)-1-[(4-chloro-1,6-dimethyl-1H-indol-2- yl)formamido]ethyl]benzenesulfonyl}acetate
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|
C23H25ClN2O6S
|
1
|
| 1 |
IC50 = 23.9 nM
|
|
|
|
CP0482898
|
US11304929, Example 01-004
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|
C23H25ClN2O5S
|
1
|
| 1 |
IC50 = 29.3 nM
|
|
|
|
CP0559195
|
US11304929, Example 05-003
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|
C25H29ClN2O5S
|
1
|
| 1 |
IC50 = 30.2 nM
|
|
|
|
CP0572182
|
US11304929, Example 02-001
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|
C22H22FN3O5S
|
1
|
| 1 |
IC50 = 32.8 nM
|
|
|
|
CP0429991
|
US11304929, Example 01-027
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|
C30H34ClN5O6S
|
1
|
| 1 |
IC50 = 34.2 nM
|
|
|
|
CP0478517
|
US11304929, Example 01-026
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|
C32H38ClN5O6S
|
1
|
| 1 |
IC50 = 35.9 nM
|
|
|
|
CP0559198
|
2-methanesulfonylethyl 2-{4-[(1R)-1-[(4-chloro-1,6-dimethyl-1H-indol-2- yl)formamido]ethyl]benzenesulfonyl}acetate
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|
C24H27ClN2O7S2
|
1
|
| 1 |
IC50 = 37.4 nM
|
|
|
|
CP0472977
|
US11304929, Example 01-009
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|
C26H27ClN4O5S
|
1
|
| 1 |
IC50 = 44.1 nM
|
|
|
|
CP0483820
|
US11304929, Example 01-029
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|
C21H22ClN3O5S
|
1
|
| 1 |
IC50 = 51.4 nM
|
|
|
|
CP0551979
|
US11304929, Example 01-012
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|
C22H23ClN2O5S
|
1
|
| 1 |
IC50 = 52.5 nM
|
|
|
|
CP0571878
|
2-(2-ethoxyethoxy)ethyl 2-{4-[(1R)-1-[(4-chloro-1,6-dimethyl-1H-indol-2- yl)formamido]ethyl]benzenesulfonyl}acetate
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|
C27H33ClN2O7S
|
1
|
| 1 |
IC50 = 53.8 nM
|
|
|
|
CP0531727
|
US11304929, Example 02-004
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|
C23H24FN3O5S
|
1
|
| 1 |
IC50 = 62.1 nM
|
|
|
|
CP0901478
|
ethyl 2-{4-[(1R)-1-{[3-(1H-indol-7-yl)-1-methyl-1H-pyrazol-5-yl]formamido}ethyl]benzenesulfonyl}acetate
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|
C25H26N4O5S
|
1
|
| 1 |
IC50 = 64.8 nM
|
|
|
|
CP0910385
|
propan-2-yl 2-{4-[(1R)-1-[(4-chloro-1,6-dimethyl-1H-indol-2-yl)formamido]ethyl]benzenesulfonyl}acetate
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|
C24H27ClN2O5S
|
1
|
| 1 |
IC50 = 66.3 nM
|
|
|
|
CP0482899
|
US11304929, Example 02-008
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|
C24H26FN3O5S
|
1
|
| 1 |
IC50 = 68.4 nM
|
|
|
|
CP0559196
|
2-(acetyloxy)ethyl 2-{4-[(1R)-1-[(4-chloro-1,6-dimethyl-1H-indol-2- yl)formamido]ethyl]benzenesulfonyl}acetate
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|
C25H27ClN2O7S
|
1
|
| 1 |
IC50 = 69 nM
|
|
|
|
CP0559197
|
2-methylpropyl 2-{4-[(1R)-1-[(4-chloro-1,6-dimethyl-1H-indol-2- yl)formamido]ethyl]benzenesulfonyl}acetate
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|
C25H29ClN2O5S
|
1
|
| 1 |
IC50 = 70.1 nM
|
|
|
|
CP0483821
|
US11304929, Example 01-016
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|
C22H23Cl2N3O5S
|
1
|
| 1 |
IC50 = 72.1 nM
|
|
|
|
CP0910387
|
ethyl 2-{4-[(1R)-1-{[3-(1H-indazol-1-yl)-1-methyl-1H-pyrazol-5-yl]formamido}ethyl]benzenesulfonyl}acetate
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|
C24H25N5O5S
|
1
|
| 1 |
IC50 = 73.3 nM
|
|
|
|
CP0482901
|
(2S)-2-methoxypropyl 2-{4-[(1R)-1-[(4-chloro-1,6-dimethyl-1H-indol-2- yl)formamido]ethyl]benzenesulfonyl}acetate
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|
C25H29ClN2O6S
|
1
|
| 1 |
IC50 = 78.6 nM
|
|
|
|
CP0495790
|
2-methoxyethyl 2-{4-[(1R)-1-({4,5-dichloro-1,6-dimethyl-1H-pyrrolo[2,3- b]pyridin-2-yl}formamido)ethyl]benzenesulfonyl}acetate
Show/Hide
|
C23H25Cl2N3O6S
|
1
|
| 1 |
IC50 = 82.8 nM
|
|
|
|
CP0490653
|
US11304929, Example 01-006
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|
C21H21Cl2N3O5S
|
1
|
| 1 |
IC50 = 88.8 nM
|
|
|
|
CP0468812
|
(3-methyloxetan-3-yl)methyl 2-{4-[(1R)-1-{[3-(4-fluorophenyl)-1-methyl-1H- pyrazol-5-yl]formamido}ethyl]benzenesulfonyl}acetate
Show/Hide
|
C26H28FN3O6S
|
1
|
| 1 |
IC50 = 102.9 nM
|
|
|
|
CP0451162
|
US11304929, Example 01-003
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|
C25H25ClN4O5S
|
1
|
| 1 |
IC50 = 109.2 nM
|
|
|
|
CP0568563
|
US11304929, Example 02-011
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|
C24H27N3O5S
|
1
|
| 1 |
IC50 = 134.9 nM
|
|
|
|
CP0944939
|
4-chloro-N-[(1R)-1-{4-[(hydroxycarbamoyl)methanesulfonyl]phenyl}ethyl]-1,6-dimethyl-1H-indole-2-carboxamide
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|
C21H22ClN3O5S
|
1
|
| 1 |
IC50 = 135.7 nM
|
|
|
|
CP0483822
|
2-(2-hydroxyethoxy)ethyl 2-{4-[(1R)-1-[(4-chloro-1,6-dimethyl-1H-indol-2- yl)formamido]ethyl]benzenesulfonyl}acetate
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|
C25H29ClN2O7S
|
1
|
| 1 |
IC50 = 138.7 nM
|
|
|
|
CP0559679
|
2-methoxyethyl 2-{4-[(1R)-1-({4,5-dichloro-1,6-dimethyl-1H-pyrrolo[2,3- b]pyridin-2-yl}formamido)ethyl]benzenesulfonyl}-2-methylpropanoate
Show/Hide
|
C25H29Cl2N3O6S
|
1
|
| 1 |
IC50 = 141.8 nM
|
|
|
|
CP0540682
|
US11304929, Example 05-013
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|
C24H27ClN2O5S
|
1
|
| 1 |
IC50 = 165.9 nM
|
|
|
|
CP0549691
|
US11304929, Example 02-007
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|
C22H23N3O6S
|
1
|
| 1 |
IC50 = 166.6 nM
|
|
|
|
CP0423638
|
2-[4-[(1S)-1-[(4,5-dichloro-1,6-dimethylindole-2-carbonyl)amino]-2-hydroxyethyl]phenyl]sulfonylacetic acid
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|
C21H20Cl2N2O6S
|
1
|
| 1 |
IC50 = 203.3 nM
|
|
|
|
CP0910389
|
2-[(2-{4-[(1R)-1-[(4-chloro-1,6-dimethyl-1H-indol-2-yl)formamido]ethyl]benzenesulfonyl}acetyl)oxy]ethyl2-{4-[(1R)-1-[(4-chloro-1,6-dimethyl-1H-indol-2-yl)formamido]ethyl]benzenesulfonyl}acetate
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|
C44H44Cl2N4O10S2
|
1
|
| 1 |
IC50 = 249 nM
|
|
|
|
CP0909714
|
ethyl 2-{4-[(1R)-1-{[3-(1H-indol-1-yl)-1-methyl-1H-pyrazol-5-yl]formamido}ethyl]benzenesulfonyl}acetate
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|
C25H26N4O5S
|
1
|
| 1 |
IC50 = 309.2 nM
|
|
|
|
CP0529474
|
US11304929, Example 01-011
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|
C27H29ClN4O5S
|
1
|
| 1 |
IC50 = 489.3 nM
|
|
|
|
CP0478518
|
US11304929, Example 05-019
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|
C24H25ClN2O5S
|
1
|
| 1 |
IC50 = 508.8 nM
|
|
|
|
CP0559678
|
US11304929, Example 02-010
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|
C21H22N4O5S
|
1
|
| 1 |
IC50 = 593.7 nM
|
|
|
|
CP0472978
|
US11304929, Example 05-005
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|
C25H29ClN2O6S
|
1
|
| 1 |
IC50 = 831.2 nM
|
|
|
|
CP0577148
|
US11304929, Example 05-001
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|
C26H31ClN2O5S
|
1
|
| 1 |
IC50 = 891.4 nM
|
|
|
|
CP0571877
|
US11304929, Example 05-012
Show/Hide
|
C26H31ClN2O5S
|
1
|
| 1 |
IC50 = 906.1 nM
|
|
|
|
CP0238143
|
2-[4-[(1R)-1-[(4,5-dichloro-1,6-dimethylindole-2-carbonyl)amino]ethyl]phenyl]sulfonylacetic acid
Show/Hide
|
C21H20Cl2N2O5S
|
1
|
| 1 |
IC50 = 1068.1 nM
|
|
|
|
CP0477290
|
2-{4-[(1R)-1-[(4-chloro-1,6-dimethyl-1H-indol-2- yl)formamido]ethyl]benzenesulfonyl}-2-methylpropanoic acid
Show/Hide
|
C23H25ClN2O5S
|
1
|
| 1 |
IC50 = 1187.5 nM
|
|
|
|
CP0969170
|
ethyl 2-{4-[(1R)-1-[(1-methyl-5-phenyl-1H-pyrazol-3-yl)formamido]ethyl]benzenesulfonyl}acetate
Show/Hide
|
C23H25N3O5S
|
1
|
| 1 |
IC50 = 1303.4 nM
|
|
|
|
CP0571876
|
2-{4-[(1S)-1-[(4-chloro-1,6-dimethyl-1H-indol-2-yl)formamido]-2- hydroxyethyl]benzenesulfonyl}acetic acid
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|
C21H21ClN2O6S
|
1
|
| 1 |
IC50 = 1377 nM
|
|
|
|
CP0551987
|
US11304929, Example 06-002
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|
C24H26FN3O5S
|
1
|
| 1 |
IC50 = 1884 nM
|
|
|
|
CP0551984
|
2-{4-[(1S)-1-({4,5-dichloro-1,6-dimethyl-1H-pyrrolo[2,3-b]pyridin-2- yl}formamido)-2-hydroxyethyl]benzenesulfonyl}acetic acid
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|
C20H19Cl2N3O6S
|
1
|
| 1 |
IC50 = 1998 nM
|
|
|
|
CP0529473
|
2-{4-[(1R)-1-[(4-chloro-1,6-dimethyl-1H-indol-2- yl)formamido]ethyl]benzenesulfonyl}pentanoic acid
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|
C24H27ClN2O5S
|
1
|
| 1 |
IC50 = 2392.2 nM
|
|
|
|
CP0961557
|
N-[(1R)-1-[4-(1-carbamoyl-1-methylethanesulfonyl)phenyl]ethyl]-4-chloro-1,6-dimethyl-1H-indole-2-carboxamide
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|
C23H26ClN3O4S
|
1
|
| 1 |
IC50 = 3216.7 nM
|
|
|
|
CP0944949
|
4-chloro-N-[(1R)-1-{4-[(dimethylcarbamoyl)methanesulfonyl]phenyl}ethyl]-1,6-dimethyl-1H-indole-2-carboxamide
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|
C23H26ClN3O4S
|
1
|
| 1 |
IC50 = 3392.1 nM
|
|
|
|
CP0483819
|
2-[4-[(1R)-1-[(4-chloro-1,6-dimethylindole-2-carbonyl)amino]ethyl]phenyl]sulfonylacetic acid
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|
C21H21ClN2O5S
|
1
|
| 1 |
IC50 = 3567.9 nM
|
|
|
|
CP0903544
|
3-(4-fluorophenyl)-N-[(1R)-1-{4-[(methoxycarbamoyl)methanesulfonyl]phenyl}ethyl]-1-methyl-1H-pyrazole-5-carboxamide
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|
C22H23FN4O5S
|
1
|
| 1 |
IC50 = 6273.5 nM
|
|
|
|
CP0534940
|
4-{4-[(1R)-1-[(4-chloro-1,6-dimethyl-1H-indol-2- yl)formamido]ethyl]benzenesulfonyl}oxane-4-carboxylic acid
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|
C25H27ClN2O6S
|
1
|
| 1 |
IC50 = 6902.8 nM
|
|
|
|
CP0883916
|
5-{4-[(1R)-1-[(4-chloro-1,6-dimethyl-1H-indol-2-yl)formamido]ethyl]benzenesulfonyl}-4-oxopentanoic acid
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|
C24H25ClN2O6S
|
1
|
| 1 |
IC50 = 9638 nM
|
|
|
|
CP0482527
|
US11304929, Example 06-001
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|
C26H28FN3O6S
|
1
|
| 1 |
IC50 = 25382.5 nM
|
|
|
|
CP0910386
|
3-(4-fluorophenyl)-1-methyl-N-[(1R)-1-[4-({[2-(morpholin-4-yl)ethoxy]carbamoyl}methanesulfonyl)phenyl]ethyl]-1H-pyrazole-5-carboxamide
Show/Hide
|
C27H32FN5O6S
|
1
|
| 1 |
IC50 = 55358.7 nM
|
|
|
|
CP0955474
|
3-(4-fluorophenyl)-1-methyl-N-[(1R)-1-[4-({[(1-methylpiperidin-4-yl)oxy]carbamoyl}methanesulfonyl)phenyl]ethyl]-1H-pyrazole-5-carboxamide
Show/Hide
|
C27H32FN5O5S
|
1
|
| 1 |
IC50 = 85293.7 nM
|
|
|
