Brief Information of the Cell Line and Protein
Cell Line ID: CL000043 , U2OS
Synonyms
U-2 OS
U-2OS
U-2-OS
U2-OS
U20-S
U20S
2T
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0042
Protein ID: PT04427 , Free fatty acid receptor 4
Gene Name FFAR4
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID Q5NUL3
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000043  Protein ID: PT04427
 
Compound ID Compound Name Compound Formula
CP0023295
(9Z,12Z)-octadeca-9,12-dienoic acid
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C18H32O2
 1
1
EC50 = 316.23 nM
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CP0463562
N-(2,4,6-trimethylphenyl)-2,3-dihydro-1,4-benzodioxine-6-sulfonamide
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C17H19NO4S
 1
1
EC50 = 316.23 nM
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CP0555634
N-(2,6-dimethyl-4-prop-2-enylphenyl)-4-methoxybenzenesulfonamide
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C18H21NO3S
 1
1
EC50 = 316.23 nM
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CP0488382
4-propyl-N-(2,4,6-trimethylphenyl)benzenesulfonamide
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C18H23NO2S
 1
1
EC50 = 398.11 nM
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CP0555633
4-methoxy-N-(4-methoxy-2,6-dimethylphenyl)benzenesulfonamide
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C16H19NO4S
 1
1
EC50 = 398.11 nM
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CP0006743
4-methoxy-N-(2,4,6-trimethylphenyl)benzenesulfonamide
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C16H19NO3S
 1
1
EC50 = 501.19 nM
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CP0481934
N-(4-chloro-2,6-dimethylphenyl)-4-methoxybenzenesulfonamide
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C15H16ClNO3S
 1
1
EC50 = 501.19 nM
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CP0411326
4-chloro-3-methoxy-N-(2,4,6-trimethylphenyl)benzenesulfonamide
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C16H18ClNO3S
 1
1
EC50 = 794.33 nM
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CP0379888
CA inhibitor, 4
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C16H19NO2S
 1
1
EC50 = 1000 nM
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CP0555632
N-(4-fluoro-2,6-dimethylphenyl)-4-methoxybenzenesulfonamide
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C15H16FNO3S
 1
1
EC50 = 1000 nM
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CP0553455
4-(trifluoromethoxy)-N-(2,4,6-trimethylphenyl)benzenesulfonamide
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C16H16F3NO3S
 1
1
EC50 = 1258.93 nM
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CP0379672
4-propan-2-yloxy-N-(2,4,6-trimethylphenyl)benzenesulfonamide
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C18H23NO3S
 1
1
EC50 = 1995.26 nM
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CP0379927
N-(2,4,6-trimethylphenyl)-3,4-dihydro-2H-1,5-benzodioxepine-7-sulfonamide
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C18H21NO4S
 1
1
EC50 = 1995.26 nM
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CP0379891
N-(2,4-dimethylphenyl)-4-methoxybenzenesulfonamide
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C15H17NO3S
 1
1
EC50 = 2511.89 nM
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CP0411806
4-chloro-N-(2,4,6-trimethylphenyl)benzenesulfonamide
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C15H16ClNO2S
 1
1
EC50 = 3162.28 nM
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CP0463452
N-(2,6-dimethylphenyl)-4-methoxybenzenesulfonamide
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C15H17NO3S
 1
1
EC50 = 3162.28 nM
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CP0414164
methyl 2-methyl-3-[(4-methylphenyl)sulfonylamino]benzoate
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C16H17NO4S
 1
1
EC50 = 3981.07 nM
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CP0494507
4-fluoro-N-(2,4,6-trimethylphenyl)benzenesulfonamide
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C15H16FNO2S
 1
1
EC50 = 6309.57 nM
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CP0411324
4-acetyl-N-(2,4,6-trimethylphenyl)benzenesulfonamide
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C17H19NO3S
 1
1
EC50 = 7943.28 nM
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CP0411898
3,4-dimethoxy-N-(2,4,6-trimethylphenyl)benzenesulfonamide
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C17H21NO4S
 1
1
EC50 = 10000 nM
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CP0411805
N-(2,4,6-trimethylphenyl)benzenesulfonamide
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C15H17NO2S
 1
1
EC50 = 12589.25 nM
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CP0536621
3-methoxy-N-(2,4,6-trimethylphenyl)benzenesulfonamide
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C16H19NO3S
 1
1
EC50 = 12589.25 nM
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CP0270777
N-(4-hydroxy-2,6-dimethylphenyl)-4-methoxybenzenesulfonamide
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C15H17NO4S
 1
1
EC50 > 31622.78 nM
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CP0379851
4-methoxy-N-(3-methylphenyl)benzenesulfonamide
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C14H15NO3S
 1
1
EC50 > 31622.78 nM
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CP0379890
4-methyl-N-(9H-xanthen-9-yl)benzenesulfonamide
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C20H17NO3S
 2
1
EC50 > 31622.78 nM
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2
IC50 = 79.43 nM
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CP0411803
4-phenyl-N-(2,4,6-trimethylphenyl)benzenesulfonamide
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C21H21NO2S
 1
1
EC50 > 31622.78 nM
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CP0419438
N-[4-(cyclopropylmethyl)-2,6-dimethylphenyl]-4-methoxybenzenesulfonamide
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C19H23NO3S
 1
1
EC50 > 31622.78 nM
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CP0419439
4-[(4-methoxyphenyl)sulfonylamino]-3,5-dimethylbenzoic acid
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C16H17NO5S
 1
1
EC50 > 31622.78 nM
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CP0419440
N-[4-(hydroxymethyl)-2,6-dimethylphenyl]-4-methoxybenzenesulfonamide
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C16H19NO4S
 1
1
EC50 > 31622.78 nM
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CP0463561
4-methoxy-N-methyl-N-(2,4,6-trimethylphenyl)benzenesulfonamide
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C17H21NO3S
 1
1
EC50 > 31622.78 nM
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CP0494492
N-(4-cyano-2,6-dimethylphenyl)-4-methoxybenzenesulfonamide
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C16H16N2O3S
 1
1
EC50 > 31622.78 nM
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CP0508187
4-methoxy-N-(4-methylphenyl)benzenesulfonamide
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C14H15NO3S
 1
1
EC50 > 31622.78 nM
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CP0520328
N-ethyl-4-methoxy-N-(2,4,6-trimethylphenyl)benzenesulfonamide
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C18H23NO3S
 1
1
EC50 > 31622.78 nM
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CP0520329
4-butoxy-N-(2,4,6-trimethylphenyl)benzenesulfonamide
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C19H25NO3S
 1
1
EC50 > 31622.78 nM
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CP0523631
4-methoxy-N-(2-methylphenyl)benzenesulfonamide
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C14H15NO3S
 1
1
EC50 > 31622.78 nM
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CP0536618
N-(2,6-diethylphenyl)-4-methoxybenzenesulfonamide
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C17H21NO3S
 1
1
EC50 > 31622.78 nM
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CP0536619
4-[(2,4,6-trimethylphenyl)sulfamoyl]benzoic acid
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C16H17NO4S
 1
1
EC50 > 31622.78 nM
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CP0536620
4-tert-butyl-N-(2,4,6-trimethylphenyl)benzenesulfonamide
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C19H25NO2S
 1
1
EC50 > 31622.78 nM
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CP0539916
methyl 4-[(4-methoxyphenyl)sulfonylamino]-3,5-dimethylbenzoate
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C17H19NO5S
 1
1
EC50 > 31622.78 nM
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CP0557735
2-methoxy-N-(2,4,6-trimethylphenyl)benzenesulfonamide
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C16H19NO3S
 1
1
EC50 > 31622.78 nM
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