Brief Information of the Cell Line and Protein
Cell Line ID: CL000852 , J-Lat 10.6
Synonyms
J-Lat clone 10.6
J-Lat full length clone 10.6
Category Cancer cell line
Organism
Homo sapiens (Human)
Protein ID: PT04279 , Protein Tat
Gene Name TAT
Organism Human immunodeficiency virus type 1 group M subtype B (isolate HXB2), HIV-1
Protein Classification Transcription factor
Uniprot ID P04608
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000852  Protein ID: PT04279
 
Compound ID Compound Name Compound Formula
CP0003580
Faridak
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C21H23N3O2
 1
1
EC50 = 130 nM
   TI
   LI
   LO
   TS
CP0085832
(1R,4S,7Z,10S,16E,21R)-7-ethylidene-4,21-di(propan-2-yl)-2-oxa-12,13-dithia-5,8,20,23-tetrazabicyclo[8.7.6]tricos-16-ene-3,6,9,19,22-pentone
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C24H36N4O6S2
 1
1
EC50 = 220 nM
   TI
   LI
   LO
   TS
CP0003832
N'-hydroxy-N-phenyloctanediamide
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C14H20N2O3
 1
1
EC50 = 2300 nM
   TI
   LI
   LO
   TS
CP0384446
4-(3-chlorophenoxy)-N-(5-cyano-1,3-thiazol-2-yl)butanamide
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C14H12ClN3O2S
 1
1
EC50 = 3100 nM
   TI
   LI
   LO
   TS
CP0253894
tert-butyl 2-[7-(4-chlorophenyl)-4,5,13-trimethyl-3-thia-1,8,11,12-tetrazatricyclo[8.3.0.02,6]trideca-2(6),4,7,10,12-pentaen-9-yl]acetate
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C23H25ClN4O2S
 1
1
EC50 = 8100 nM
   TI
   LI
   LO
   TS
CP0536736
4-[3-(trifluoromethyl)phenoxy]-N-[5-(trifluoromethyl)-1,3-thiazol-2-yl]butanamide
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C15H12F6N2O2S
 1
1
EC50 = 10000 nM
   TI
   LI
   LO
   TS
CP0479830
N-(5-cyano-1,3-thiazol-2-yl)-4-[3-(trifluoromethyl)phenoxy]butanamide
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C15H12F3N3O2S
 1
1
EC50 = 11000 nM
   TI
   LI
   LO
   TS
CP0426588
4-(5-chloropyridin-3-yl)oxy-N-(5-methyl-1,3-thiazol-2-yl)butanamide
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C13H14ClN3O2S
 1
1
EC50 = 25000 nM
   TI
   LI
   LO
   TS
CP0164338
N-(5-bromo-1,3-thiazol-2-yl)-4-(4-chloro-3-methylphenoxy)butanamide
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C14H14BrClN2O2S
 1
1
EC50 > 40000 nM
   TI
   LI
   LO
   TS
CP0368792
N-(5-methyl-1,3-thiazol-2-yl)-4-phenoxybutanamide
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C14H16N2O2S
 1
1
EC50 > 40000 nM
   TI
   LI
   LO
   TS
CP0384443
N-(5-bromo-1,3-thiazol-2-yl)-4-phenoxybutanamide
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C13H13BrN2O2S
 1
1
EC50 > 40000 nM
   TI
   LI
   LO
   TS
CP0384445
N-(5-chloro-1,3-thiazol-2-yl)-4-[3-(trifluoromethyl)phenoxy]butanamide
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C14H12ClF3N2O2S
 1
1
EC50 > 40000 nM
   TI
   LI
   LO
   TS
CP0438018
4-(4-chloro-3-methylphenoxy)-N-(5-chloro-1,3-thiazol-2-yl)butanamide
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C14H14Cl2N2O2S
 1
1
EC50 > 40000 nM
   TI
   LI
   LO
   TS
CP0440379
N-(5-cyano-1,3-thiazol-2-yl)-4-phenoxybutanamide
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C14H13N3O2S
 1
1
EC50 > 40000 nM
   TI
   LI
   LO
   TS