| Compound ID |
Compound Name |
Compound Formula |
|
CP0422038
|
N-[5-[2-amino-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-2,3-dimethoxyphenyl]propane-1-sulfonamide
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|
C26H33N5O4S
|
1
|
| 1 |
IC50 = 1 nM
|
|
|
|
CP0252329
|
N-[5-[2-amino-5-(3-piperazin-1-ylphenyl)pyridin-3-yl]-3-fluoro-2-methoxyphenyl]propane-1-sulfonamide
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|
C25H30FN5O3S
|
1
|
| 1 |
IC50 = 16 nM
|
|
|
|
CP0265170
|
N-[5-[2-amino-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-3-fluoro-2-methoxyphenyl]propane-1-sulfonamide
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|
C25H30FN5O3S
|
1
|
| 1 |
IC50 = 26 nM
|
|
|
|
CP0313144
|
N-[3-[2-amino-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-5-ethoxyphenyl]propane-2-sulfonamide
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|
C26H33N5O3S
|
1
|
| 1 |
IC50 = 46 nM
|
|
|
|
CP0363847
|
N-[5-[2-amino-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-3-chloro-2-methoxyphenyl]propane-1-sulfonamide
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|
C25H30ClN5O3S
|
1
|
| 1 |
IC50 = 46 nM
|
|
|
|
CP0490922
|
N-[3-[2-amino-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-5-methoxyphenyl]benzenesulfonamide
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|
C28H29N5O3S
|
1
|
| 1 |
IC50 = 53 nM
|
|
|
|
CP0265172
|
N-[3-[2-amino-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-5-methoxyphenyl]propane-2-sulfonamide
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|
C25H31N5O3S
|
1
|
| 1 |
IC50 = 121 nM
|
|
|
|
CP0142352
|
N-[5-[2-amino-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-2-methoxy-3-methylphenyl]propane-1-sulfonamide
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|
C26H33N5O3S
|
1
|
| 1 |
IC50 = 129 nM
|
|
|
|
CP0265171
|
N-[3-[2-amino-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-5-methoxyphenyl]propane-1-sulfonamide
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|
C25H31N5O3S
|
1
|
| 1 |
IC50 = 243 nM
|
|
|
|
CP0252328
|
N-[3-[2-amino-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-5-propan-2-yloxyphenyl]propane-2-sulfonamide
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|
C27H35N5O3S
|
1
|
| 1 |
IC50 = 323 nM
|
|
|
|
CP0534930
|
N-[3-fluoro-2-methoxy-5-[5-(4-piperazin-1-ylphenyl)pyridin-3-yl]phenyl]propane-1-sulfonamide
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|
C25H29FN4O3S
|
1
|
| 1 |
IC50 = 352 nM
|
|
|
|
CP0552860
|
N-[3-[2-amino-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-5-methoxyphenyl]methanesulfonamide
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|
C23H27N5O3S
|
1
|
| 1 |
IC50 = 390 nM
|
|
|
|
CP0142377
|
N-[5-[2-amino-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-2-methoxyphenyl]propane-1-sulfonamide
Show/Hide
|
C25H31N5O3S
|
1
|
| 1 |
IC50 = 420 nM
|
|
|
|
CP0552859
|
N-[3-methoxy-5-[2-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]phenyl]propane-2-sulfonamide
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|
C26H32N4O3S
|
1
|
| 1 |
IC50 = 523 nM
|
|
|
|
CP0357506
|
3-(3-fluoro-4,5-dimethoxyphenyl)-5-(4-piperazin-1-ylphenyl)pyridin-2-amine
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|
C23H25FN4O2
|
1
|
| 1 |
IC50 = 595 nM
|
|
|
|
CP0422149
|
2-[2-[2-[benzenesulfonyl(methyl)amino]ethyl]benzimidazol-1-yl]-N-(2,3-dihydro-1H-inden-5-yl)acetamide
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|
C27H28N4O3S
|
1
|
| 1 |
IC50 = 630 nM
|
|
|
|
CP0322297
|
5-(4-piperazin-1-ylphenyl)-3-(4-propylsulfonyl-2,3-dihydro-1,4-benzoxazin-6-yl)pyridin-2-amine
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|
C26H31N5O3S
|
1
|
| 1 |
IC50 = 1011 nM
|
|
|
|
CP0136272
|
N-[5-[2-amino-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-2-methylphenyl]propane-1-sulfonamide
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|
C25H31N5O2S
|
1
|
| 1 |
IC50 = 1064 nM
|
|
|
|
CP0534929
|
N-[[5-[2-amino-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-2-methoxyphenyl]methyl]propane-1-sulfonamide
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|
C26H33N5O3S
|
1
|
| 1 |
IC50 = 1290 nM
|
|
|
|
CP0538394
|
5-(4-piperazin-1-ylphenyl)-3-(1-propylsulfonyl-2,3-dihydroindol-6-yl)pyridin-2-amine
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|
C26H31N5O2S
|
1
|
| 1 |
IC50 = 2426 nM
|
|
|
|
CP0313147
|
N-[7-[2-amino-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-2,3-dihydro-1,4-benzodioxin-5-yl]propane-1-sulfonamide
Show/Hide
|
C26H31N5O4S
|
1
|
| 1 |
IC50 = 2458 nM
|
|
|
|
CP0565408
|
N-[3-fluoro-2-methoxy-5-[2-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]phenyl]propane-1-sulfonamide
Show/Hide
|
C26H31FN4O3S
|
1
|
| 1 |
IC50 = 2556 nM
|
|
|
|
CP0512470
|
N-[5-[2-amino-5-(3-methylsulfonylphenyl)pyridin-3-yl]-2-methoxyphenyl]propane-1-sulfonamide
Show/Hide
|
C22H25N3O5S2
|
1
|
| 1 |
IC50 = 2655 nM
|
|
|
|
CP0313148
|
N-[3-methoxy-5-[2-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]phenyl]propane-1-sulfonamide
Show/Hide
|
C26H32N4O3S
|
1
|
| 1 |
IC50 = 2669 nM
|
|
|
|
CP0313150
|
N-[2-methoxy-4-[2-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]phenyl]propane-1-sulfonamide
Show/Hide
|
C26H32N4O3S
|
1
|
| 1 |
IC50 = 2944 nM
|
|
|
|
CP0444014
|
N-[2-[1-[2-(2,3-dihydro-1H-inden-5-ylamino)-2-oxoethyl]benzimidazol-2-yl]ethyl]benzamide
Show/Hide
|
C27H26N4O2
|
2
|
| 1 |
IC50 = 3300 nM
|
|
|
| 2 |
IC50 = 6200 nM
|
|
|
|
CP0313151
|
N-[5-[2-amino-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-3-methoxy-2-methylphenyl]propane-1-sulfonamide
Show/Hide
|
C26H33N5O3S
|
1
|
| 1 |
IC50 = 3347 nM
|
|
|
|
CP0136353
|
N-[3-methoxy-5-[2-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]phenyl]methanesulfonamide
Show/Hide
|
C24H28N4O3S
|
1
|
| 1 |
IC50 = 3705 nM
|
|
|
|
CP0552399
|
2-[2-[2-(benzylamino)ethyl]benzimidazol-1-yl]-N-(2,3-dihydro-1H-inden-5-yl)acetamide
Show/Hide
|
C27H28N4O
|
1
|
| 1 |
IC50 = 4760 nM
|
|
|
|
CP0537944
|
2-[2-[3-[benzenesulfonyl(methyl)amino]propyl]benzimidazol-1-yl]-N-(2,3-dihydro-1H-inden-5-yl)acetamide
Show/Hide
|
C28H30N4O3S
|
1
|
| 1 |
IC50 = 5080 nM
|
|
|
|
CP0534935
|
2-[2-[3-(benzenesulfonamido)propyl]benzimidazol-1-yl]-N-(2,3-dihydro-1H-inden-5-yl)acetamide
Show/Hide
|
C27H28N4O3S
|
1
|
| 1 |
IC50 = 5120 nM
|
|
|
|
CP0471660
|
2-[2-[2-(benzenesulfonamido)ethyl]benzimidazol-1-yl]-N-(2,3-dihydro-1H-inden-5-yl)acetamide
Show/Hide
|
C26H26N4O3S
|
1
|
| 1 |
IC50 = 5230 nM
|
|
|
|
CP0568395
|
N-[3-methoxy-5-[2-methyl-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]phenyl]ethanesulfonamide
Show/Hide
|
C25H30N4O3S
|
1
|
| 1 |
IC50 = 5239 nM
|
|
|
|
CP0422152
|
N-[3-[1-[2-(2,3-dihydro-1H-inden-5-ylamino)-2-oxoethyl]benzimidazol-2-yl]propyl]benzamide
Show/Hide
|
C28H28N4O2
|
1
|
| 1 |
IC50 = 5700 nM
|
|
|
|
CP0487640
|
N-(2,3-dihydro-1H-inden-5-yl)-2-[2-[2-[[5-(dimethylamino)naphthalen-1-yl]sulfonylamino]ethyl]benzimidazol-1-yl]acetamide
Show/Hide
|
C32H33N5O3S
|
1
|
| 1 |
IC50 = 6200 nM
|
|
|
|
CP0552400
|
3-[1-[2-(2,3-dihydro-1H-inden-5-ylamino)-2-oxoethyl]benzimidazol-2-yl]-N-phenylpropanamide
Show/Hide
|
C27H26N4O2
|
1
|
| 1 |
IC50 = 8800 nM
|
|
|
|
CP0375351
|
4-benzyl-1-pentylbenzimidazol-2-amine
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|
C19H23N3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0375352
|
N-(1-pentylbenzimidazol-2-yl)acetamide
Show/Hide
|
C14H19N3O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0375357
|
1-pentyl-4-phenylbenzimidazol-2-amine
Show/Hide
|
C18H21N3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0375359
|
3-pentylbenzo[f]benzimidazol-2-amine
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|
C16H19N3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0400246
|
1-pentylbenzo[e]benzimidazol-2-amine
Show/Hide
|
C16H19N3
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0410599
|
1-pentyl-4-phenylmethoxybenzimidazol-2-amine
Show/Hide
|
C19H23N3O
|
1
|
| 1 |
IC50 > 10000 nM
|
|
|
|
CP0422101
|
tert-butyl 4-[2-[1-[2-(2,3-dihydro-1H-inden-5-ylamino)-2-oxoethyl]benzimidazol-2-yl]ethylcarbamoyl]piperidine-1-carboxylate
Show/Hide
|
C31H39N5O4
|
1
|
| 1 |
IC50 = 10600 nM
|
|
|
|
CP0422102
|
N-(2,3-dihydro-1H-inden-5-yl)-2-[2-[2-(pyridin-3-ylsulfonylamino)ethyl]benzimidazol-1-yl]acetamide
Show/Hide
|
C25H25N5O3S
|
1
|
| 1 |
IC50 = 16400 nM
|
|
|
|
CP0422098
|
N-(2,3-dihydro-1H-inden-5-yl)-2-[2-[2-[[5-(dimethylamino)naphthalen-1-yl]sulfonyl-methylamino]ethyl]benzimidazol-1-yl]acetamide
Show/Hide
|
C33H35N5O3S
|
1
|
| 1 |
IC50 > 20000 nM
|
|
|
|
CP0422148
|
N-(2,3-dihydro-1H-inden-5-yl)-2-[2-[2-(pyridin-4-ylmethylamino)ethyl]benzimidazol-1-yl]acetamide
Show/Hide
|
C26H27N5O
|
1
|
| 1 |
IC50 = 22900 nM
|
|
|
|
CP0565922
|
N-[2-[1-[2-(2,3-dihydro-1H-inden-5-ylamino)-2-oxoethyl]benzimidazol-2-yl]ethyl]-2-pyridin-4-ylacetamide
Show/Hide
|
C27H27N5O2
|
1
|
| 1 |
IC50 = 25900 nM
|
|
|
|
CP0552892
|
5-ethyl-N-[2-fluoro-5-(2-methyl-4-oxoquinazolin-3-yl)phenyl]thiophene-2-sulfonamide
Show/Hide
|
C21H18FN3O3S2
|
1
|
| 1 |
IC50 > 50000 nM
|
|
|
|
CP0142376
|
(1-tosylbenzimidazol-2-yl)amine
Show/Hide
|
C14H13N3O2S
|
1
|
| 1 |
IC50 = 54900 nM
|
|
|
|
CP0313145
|
N-[5-[2-amino-5-(4-piperazin-1-ylphenyl)pyridin-3-yl]-2-hydroxyphenyl]propane-1-sulfonamide
Show/Hide
|
C24H29N5O3S
|
1
|
| 1 |
IC50 > 1000 nM
|
|
|
