| Compound ID |
Compound Name |
Compound Formula |
|
CP0212474
|
1-[4-[4-[1-methyl-5-[[(1R)-1-[3-(trifluoromethyl)phenyl]ethoxy]carbonylamino]triazol-4-yl]phenyl]phenyl]cyclopropane-1-carboxylic acid
Show/Hide
|
C29H25F3N4O4
|
1
|
| 1 |
IC50 = 17 nM
|
|
|
|
CP0169579
|
1-[4-[3-fluoro-4-[1-methyl-5-[[(1R)-1-phenylethoxy]carbonylamino]triazol-4-yl]phenyl]phenyl]cyclopropane-1-carboxylic acid
Show/Hide
|
C28H25FN4O4
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0238378
|
1-[4-[4-[1-methyl-5-[[(1R)-1-phenylethoxy]carbonylamino]triazol-4-yl]phenyl]phenyl]cyclopropane-1-carboxylic acid
Show/Hide
|
C28H26N4O4
|
1
|
| 1 |
IC50 = 18 nM
|
|
|
|
CP0097125
|
[(1R)-1-phenylethyl] N-[3-methyl-5-[4-[4-[1-(methylsulfonylcarbamoyl)cyclopropyl]phenyl]phenyl]triazol-4-yl]carbamate
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|
C29H29N5O5S
|
1
|
| 1 |
IC50 = 19 nM
|
|
|
|
CP0138967
|
1-[4-[4-[1-methyl-5-[[(1R)-1-phenylethoxy]carbonylamino]pyrazol-4-yl]phenyl]phenyl]cyclopropane-1-carboxylic acid
Show/Hide
|
C29H27N3O4
|
1
|
| 1 |
IC50 = 21 nM
|
|
|
|
CP0248761
|
[(1R)-1-phenylethyl] N-[5-methyl-3-[4-[4-[1-(2H-tetrazol-5-yl)cyclopropyl]phenyl]phenyl]triazol-4-yl]carbamate
Show/Hide
|
C28H26N8O2
|
1
|
| 1 |
IC50 = 23 nM
|
|
|
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CP0169580
|
[(1R)-1-[3-(trifluoromethyl)phenyl]ethyl] N-[3-methyl-5-[4-[4-[1-(methylsulfonylcarbamoyl)cyclopropyl]phenyl]phenyl]triazol-4-yl]carbamate
Show/Hide
|
C30H28F3N5O5S
|
1
|
| 1 |
IC50 = 24 nM
|
|
|
|
CP0282928
|
1-[4-[4-[5-[[(1R)-1-(2-fluorophenyl)ethoxy]carbonylamino]-1-methylpyrazol-4-yl]phenyl]phenyl]cyclopropane-1-carboxylic acid
Show/Hide
|
C29H26FN3O4
|
1
|
| 1 |
IC50 = 24 nM
|
|
|
|
CP0282929
|
1-[4-[4-[4-methyl-5-[[(1R)-1-phenylethoxy]carbonylamino]triazol-1-yl]phenyl]phenyl]cyclopropane-1-carboxylic acid
Show/Hide
|
C28H26N4O4
|
1
|
| 1 |
IC50 = 25.2 nM
|
|
|
|
CP0169578
|
[(1R)-1-phenylethyl] N-[5-methyl-3-[4-[4-[1-(methylsulfonylcarbamoyl)cyclopropyl]phenyl]phenyl]triazol-4-yl]carbamate
Show/Hide
|
C29H29N5O5S
|
1
|
| 1 |
IC50 = 32 nM
|
|
|
|
CP0212472
|
1-[4-[4-[5-[[(1R)-1-(2-fluorophenyl)ethoxy]carbonylamino]-4-methyltriazol-1-yl]phenyl]phenyl]cyclopropane-1-carboxylic acid
Show/Hide
|
C28H25FN4O4
|
1
|
| 1 |
IC50 = 34.5 nM
|
|
|
|
CP0282927
|
2-[4-[4-[1-methyl-5-[[(1R)-1-phenylethoxy]carbonylamino]pyrazol-4-yl]phenyl]phenyl]acetic acid
Show/Hide
|
C27H25N3O4
|
1
|
| 1 |
IC50 = 35 nM
|
|
|
|
CP0315964
|
1-[4-[4-[5-[[(1R)-1-phenylethoxy]carbonylamino]triazol-1-yl]phenyl]phenyl]cyclopropane-1-carboxylic acid
Show/Hide
|
C27H24N4O4
|
1
|
| 1 |
IC50 = 36 nM
|
|
|
|
CP0342652
|
1-[4-[4-[5-[[(2R)-butan-2-yl]oxycarbonylamino]-1-methylpyrazol-4-yl]phenyl]phenyl]cyclopropane-1-carboxylic acid
Show/Hide
|
C25H27N3O4
|
1
|
| 1 |
IC50 = 38 nM
|
|
|
|
CP0193811
|
1-[4-[4-[1-methyl-5-[[(1R)-1-[3-(trifluoromethyl)phenyl]ethoxy]carbonylamino]pyrazol-4-yl]phenyl]phenyl]cyclopropane-1-carboxylic acid
Show/Hide
|
C30H26F3N3O4
|
1
|
| 1 |
IC50 = 41 nM
|
|
|
|
CP0212473
|
1-[4-[4-[4-ethyl-5-[[(1R)-1-phenylethoxy]carbonylamino]triazol-1-yl]phenyl]phenyl]cyclopropane-1-carboxylic acid
Show/Hide
|
C29H28N4O4
|
1
|
| 1 |
IC50 = 42 nM
|
|
|
|
CP0323007
|
2-[4-[4-[1-methyl-5-[[(1R)-1-phenylethoxy]carbonylamino]triazol-4-yl]phenyl]phenyl]acetic acid
Show/Hide
|
C26H24N4O4
|
1
|
| 1 |
IC50 = 48 nM
|
|
|
|
CP0193810
|
1-[4-[4-[5-[1-(4-fluorophenyl)ethoxycarbonylamino]-1-methylpyrazol-4-yl]phenyl]phenyl]cyclopropane-1-carboxylic acid
Show/Hide
|
C29H26FN3O4
|
1
|
| 1 |
IC50 = 57 nM
|
|
|
|
CP0212475
|
2-[4-[4-[1-methyl-5-[[(1R)-1-phenylethoxy]carbonylamino]triazol-4-yl]phenyl]cyclohexyl]acetic acid
Show/Hide
|
C26H30N4O4
|
1
|
| 1 |
IC50 = 58 nM
|
|
|
|
CP0193813
|
1-[4-[4-[1-methyl-5-[[(2R)-3-methylbutan-2-yl]oxycarbonylamino]triazol-4-yl]phenyl]phenyl]cyclopropane-1-carboxylic acid
Show/Hide
|
C25H28N4O4
|
1
|
| 1 |
IC50 = 70 nM
|
|
|
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CP0378587
|
5-amino-1-[N-cyclopentyl-C-(2-fluoro-4-methoxybenzoyl)carbonimidoyl]pyrazole-4-carbonitrile
Show/Hide
|
C18H18FN5O2
|
1
|
| 1 |
IC50 = 74 nM
|
|
|
|
CP0487523
|
5-amino-1-[N-cyclopentyl-C-(2,4-dimethoxybenzoyl)carbonimidoyl]pyrazole-4-carbonitrile
Show/Hide
|
C19H21N5O3
|
1
|
| 1 |
IC50 = 79 nM
|
|
|
|
CP0238376
|
1-[4-[4-[1-methyl-5-[[(2R)-3-methylbutan-2-yl]oxycarbonylamino]pyrazol-4-yl]phenyl]phenyl]cyclopropane-1-carboxylic acid
Show/Hide
|
C26H29N3O4
|
1
|
| 1 |
IC50 = 106 nM
|
|
|
|
CP0553563
|
5-amino-1-[C-(2,4-dimethoxybenzoyl)-N-propan-2-ylcarbonimidoyl]pyrazole-4-carbonitrile
Show/Hide
|
C17H19N5O3
|
1
|
| 1 |
IC50 = 111 nM
|
|
|
|
CP0138968
|
1-[4-[4-[4-methyl-5-[[(1R)-1-[2-(trifluoromethyl)phenyl]ethoxy]carbonylamino]triazol-1-yl]phenyl]phenyl]cyclopropane-1-carboxylic acid
Show/Hide
|
C29H25F3N4O4
|
1
|
| 1 |
IC50 = 112 nM
|
|
|
|
CP0169577
|
1-[4-[4-[5-(1-cyclobutylethoxycarbonylamino)-4-methyltriazol-1-yl]phenyl]phenyl]cyclopropane-1-carboxylic acid
Show/Hide
|
C26H28N4O4
|
1
|
| 1 |
IC50 = 161 nM
|
|
|
|
CP0342653
|
1-[4-[4-[4-methyl-5-[[(1R)-1-[3-(trifluoromethyl)phenyl]ethoxy]carbonylamino]triazol-1-yl]phenyl]phenyl]cyclopropane-1-carboxylic acid
Show/Hide
|
C29H25F3N4O4
|
1
|
| 1 |
IC50 = 174 nM
|
|
|
|
CP0103368
|
1-[4-[4-[5-(cyclobutyloxycarbonylamino)-1-methylpyrazol-4-yl]phenyl]phenyl]cyclopropane-1-carboxylic acid
Show/Hide
|
C25H25N3O4
|
1
|
| 1 |
IC50 = 176 nM
|
|
|
|
CP0449672
|
1-[4-[4-[4-methyl-5-[[(2R)-3-methylbutan-2-yl]oxycarbonylamino]triazol-1-yl]phenyl]phenyl]cyclopropane-1-carboxylic acid
Show/Hide
|
C25H28N4O4
|
1
|
| 1 |
IC50 = 217 nM
|
|
|
|
CP0193812
|
1-[4-[4-[5-[[(2R)-butan-2-yl]oxycarbonylamino]-4-methyltriazol-1-yl]phenyl]phenyl]cyclopropane-1-carboxylic acid
Show/Hide
|
C24H26N4O4
|
1
|
| 1 |
IC50 = 398 nM
|
|
|
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CP0480326
|
5-amino-1-[N-cyclohexyl-C-(2,4-dimethoxybenzoyl)carbonimidoyl]pyrazole-4-carbonitrile
Show/Hide
|
C20H23N5O3
|
1
|
| 1 |
IC50 = 510 nM
|
|
|
|
CP0510299
|
5-amino-1-[N-cyclopentyl-C-(4-ethylbenzoyl)carbonimidoyl]pyrazole-4-carbonitrile
Show/Hide
|
C19H21N5O
|
1
|
| 1 |
IC50 = 586 nM
|
|
|
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CP0342651
|
[(1R)-1-(2-chlorophenyl)ethyl] N-[4-(2-fluorophenyl)-2-methylpyrazol-3-yl]carbamate
Show/Hide
|
C19H17ClFN3O2
|
1
|
| 1 |
IC50 = 644 nM
|
|
|
|
CP0508666
|
5-amino-1-[N-cyclopentyl-C-(3-methoxynaphthalene-2-carbonyl)carbonimidoyl]pyrazole-4-carbonitrile
Show/Hide
|
C22H21N5O2
|
1
|
| 1 |
IC50 = 805 nM
|
|
|
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CP0463420
|
5-amino-1-[N-cyclopentyl-C-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)carbonimidoyl]pyrazole-4-carbonitrile
Show/Hide
|
C21H23N5O2
|
1
|
| 1 |
IC50 = 825 nM
|
|
|
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CP0085018
|
1-[4-[4-[4-methyl-5-[(2-methylpropan-2-yl)oxycarbonylamino]triazol-1-yl]phenyl]phenyl]cyclopropane-1-carboxylic acid
Show/Hide
|
C24H26N4O4
|
1
|
| 1 |
IC50 = 985 nM
|
|
|
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CP0241461
|
1-[4-[4-[1-methyl-5-[[(1S)-1-[3-(trifluoromethyl)phenyl]ethoxy]carbonylamino]triazol-4-yl]phenyl]phenyl]cyclopropane-1-carboxylic acid
Show/Hide
|
C29H25F3N4O4
|
1
|
| 1 |
IC50 = 2650 nM
|
|
|
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CP0480354
|
5-amino-1-[C-(4-bromobenzoyl)-N-cyclopentylcarbonimidoyl]pyrazole-4-carbonitrile
Show/Hide
|
C17H16BrN5O
|
1
|
| 1 |
IC50 = 2940 nM
|
|
|
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CP0510300
|
5-amino-1-[N-cyclopentyl-C-(2,4,5-trimethoxybenzoyl)carbonimidoyl]pyrazole-4-carbonitrile
Show/Hide
|
C20H23N5O4
|
1
|
| 1 |
IC50 = 3358 nM
|
|
|
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CP0169576
|
1-(2-chlorophenyl)ethyl N-(2-methyl-4-phenylpyrazol-3-yl)carbamate
Show/Hide
|
C19H18ClN3O2
|
1
|
| 1 |
IC50 = 3590 nM
|
|
|
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CP0238372
|
1-(2-chlorophenyl)ethyl N-[4-(4-fluorophenyl)-2-methylpyrazol-3-yl]carbamate
Show/Hide
|
C19H17ClFN3O2
|
1
|
| 1 |
IC50 = 3970 nM
|
|
|
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CP0212478
|
[(1R)-1-phenylethyl] N-(2-methyl-4-phenylpyrazol-3-yl)carbamate
Show/Hide
|
C19H19N3O2
|
1
|
| 1 |
IC50 = 17500 nM
|
|
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CP0085016
|
[(1R)-1-phenylethyl] N-[4-(4-methoxyphenyl)-2-methylpyrazol-3-yl]carbamate
Show/Hide
|
C20H21N3O3
|
1
|
| 1 |
IC50 > 30000 nM
|
|
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CP0212471
|
[(1R)-1-phenylethyl] N-[2-methyl-4-(4-phenylphenyl)pyrazol-3-yl]carbamate
Show/Hide
|
C25H23N3O2
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
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CP0238374
|
[(1S)-1-(2-chlorophenyl)ethyl] N-[4-(2-fluorophenyl)-2-methylpyrazol-3-yl]carbamate
Show/Hide
|
C19H17ClFN3O2
|
1
|
| 1 |
IC50 > 30000 nM
|
|
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CP0238375
|
2-[4-[1-methyl-5-[[(1R)-1-phenylethoxy]carbonylamino]pyrazol-4-yl]phenyl]acetic acid
Show/Hide
|
C21H21N3O4
|
1
|
| 1 |
IC50 > 30000 nM
|
|
|
