Compound ID |
Compound Name |
Compound Formula |
CP0477581
|
3-[1-[(2S,3S)-2-(2,3-dihydro-1H-inden-2-ylmethyl)-3-(3,5-dimethoxy-4-methylphenyl)-3-hydroxypropyl]pyrrol-3-yl]propanoic acid
Show/Hide
|
C29H35NO5
|
3
|
1 |
IC50 = 0.16 nM
|
|
|
2 |
IC50 = 0.19 nM
|
|
|
3 |
IC50 = 86 nM
|
|
|
CP0089898
|
5-chloro-2-[4-[[(3,5-dimethoxy-4-methylbenzoyl)-(3-phenylpropyl)amino]methyl]phenoxy]benzoic acid
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|
C33H32ClNO6
|
1
|
1 |
IC50 = 3.5 nM
|
|
|
CP0576287
|
(1S,3S)-3-[6-[3-methyl-4-[(2-phenylethylsulfonylamino)methyl]-1,2-oxazol-5-yl]pyridin-3-yl]oxycyclohexane-1-carboxylic acid
Show/Hide
|
C25H29N3O6S
|
1
|
1 |
IC50 = 4 nM
|
|
|
CP0459357
|
(1S,3S)-3-[6-[4-[[(3-fluorophenyl)methoxycarbonylamino]methyl]-3-methyl-1,2-oxazol-5-yl]pyridin-3-yl]oxycyclohexane-1-carboxylic acid
Show/Hide
|
C25H26FN3O6
|
1
|
1 |
IC50 = 5 nM
|
|
|
CP0543033
|
4-chloro-2-[4-[[(3,5-dimethoxy-4-methylbenzoyl)-(3-phenylpropyl)amino]methyl]phenoxy]benzoic acid
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|
C33H32ClNO6
|
1
|
1 |
IC50 = 5.9 nM
|
|
|
CP0952861
|
(R)-2-((2-(2-fluoro-4-methoxyphenyl)-2-hydroxy-N-(3-phenylpropyl)acetamido)methyl)-5-methyl-N-(methylsulfonyl)thiazole-4-carboxamide
Show/Hide
|
C25H28FN3O6S2
|
1
|
1 |
IC50 = 6.6 nM
|
|
|
CP0558533
|
(1S,3S)-3-[6-[4-[[(4-fluorophenyl)methoxycarbonylamino]methyl]-3-methyl-1,2-oxazol-5-yl]pyridin-3-yl]oxycyclohexane-1-carboxylic acid
Show/Hide
|
C25H26FN3O6
|
1
|
1 |
IC50 = 9 nM
|
|
|
CP0384713
|
2-[1-[(2S)-2-[(S)-(3,5-dimethoxy-4-methylphenyl)-hydroxymethyl]-5-phenylpentyl]pyrrol-3-yl]acetic acid
Show/Hide
|
C27H33NO5
|
1
|
1 |
IC50 = 13 nM
|
|
|
CP0530979
|
2-[4-[[(3,5-dimethoxy-4-methylbenzoyl)-(3-phenylpropyl)amino]methyl]phenoxy]-4-methylbenzoic acid
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|
C34H35NO6
|
1
|
1 |
IC50 = 15 nM
|
|
|
CP0855804
|
(R)-2-(4'-(4-((1-(2-chlorophenyl)ethoxy)carbonylamino)-3-methylisoxazol-5-yl)biphenyl-4-yl)acetic acid
Show/Hide
|
C27H23ClN2O5
|
1
|
1 |
IC50 = 17 nM
|
|
|
CP0431765
|
3-[1-[(2S)-2-[(S)-(3,5-dimethoxy-4-methylphenyl)-hydroxymethyl]-5-phenylpentyl]pyrrol-3-yl]propanoic acid
Show/Hide
|
C28H35NO5
|
1
|
1 |
IC50 = 22 nM
|
|
|
CP0477577
|
2-[1-[(2S)-2-[(S)-(3,5-dimethoxy-4-methylphenyl)-hydroxymethyl]-5-thiophen-3-ylpentyl]pyrrol-3-yl]acetic acid
Show/Hide
|
C25H31NO5S
|
1
|
1 |
IC50 = 23 nM
|
|
|
CP0148963
|
2-[4-[4-[3-methyl-4-[[(1R)-1-phenylethoxy]carbonylamino]-1,2-oxazol-5-yl]phenyl]phenyl]acetic acid
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|
C27H24N2O5
|
1
|
1 |
IC50 = 25 nM
|
|
|
CP0562327
|
(1S,3S)-3-[6-[4-[[(3,5-difluorophenyl)methoxycarbonylamino]methyl]-3-methyl-1,2-oxazol-5-yl]pyridin-3-yl]oxycyclohexane-1-carboxylic acid
Show/Hide
|
C25H25F2N3O6
|
1
|
1 |
IC50 = 27 nM
|
|
|
CP0567433
|
2-[1-[(2S)-2-[(S)-(3,5-dimethoxy-4-methylphenyl)-hydroxymethyl]-5-thiophen-2-ylpentyl]pyrrol-3-yl]acetic acid
Show/Hide
|
C25H31NO5S
|
1
|
1 |
IC50 = 29 nM
|
|
|
CP0561828
|
2-[1-[(2S)-2-[(S)-(3,5-dimethoxy-4-methylphenyl)-hydroxymethyl]-5-phenylpentyl]pyrazol-4-yl]acetic acid
Show/Hide
|
C26H32N2O5
|
1
|
1 |
IC50 = 30 nM
|
|
|
CP0536861
|
2-[1-[(2S)-2-[(S)-(3,5-dimethoxy-4-methylphenyl)-hydroxymethyl]-5-phenylpentyl]pyrazol-3-yl]acetic acid
Show/Hide
|
C26H32N2O5
|
1
|
1 |
IC50 = 32 nM
|
|
|
CP0567261
|
3-[1-[(2S)-2-[(S)-(3,5-dimethoxy-4-methylphenyl)-hydroxymethyl]-5-phenylpentyl]pyrazol-4-yl]propanoic acid
Show/Hide
|
C27H34N2O5
|
1
|
1 |
IC50 = 34 nM
|
|
|
CP0561827
|
3-[1-[(2S)-2-[(S)-(3,5-dimethoxy-4-methylphenyl)-hydroxymethyl]-5-thiophen-3-ylpentyl]pyrrol-3-yl]propanoic acid
Show/Hide
|
C26H33NO5S
|
1
|
1 |
IC50 = 38 nM
|
|
|
CP0477578
|
3-[1-[(2S)-2-[(S)-(3,5-dimethoxy-4-methylphenyl)-hydroxymethyl]-5-phenylpentyl]pyrazol-3-yl]propanoic acid
Show/Hide
|
C27H34N2O5
|
1
|
1 |
IC50 = 40 nM
|
|
|
CP0445816
|
2-[4-[[(3,5-dimethoxy-4-methylbenzoyl)-(3-phenylpropyl)amino]methyl]phenoxy]-5-methylbenzoic acid
Show/Hide
|
C34H35NO6
|
1
|
1 |
IC50 = 42 nM
|
|
|
CP0431764
|
3-[1-[(2S)-2-[(S)-(3,5-dimethoxy-4-methylphenyl)-hydroxymethyl]-5-thiophen-2-ylpentyl]pyrrol-3-yl]propanoic acid
Show/Hide
|
C26H33NO5S
|
1
|
1 |
IC50 = 45 nM
|
|
|
CP0861029
|
(R)-2-(4'-(4-((1-(2-chlorophenyl)ethoxy)carbonylamino)-3-methylisothiazol-5-yl)biphenyl-4-yl)acetic acid
Show/Hide
|
C27H23ClN2O4S
|
1
|
1 |
IC50 < 50 nM
|
|
|
CP0477576
|
2-[1-[(2S,3S)-2-(2,3-dihydro-1H-inden-2-ylmethyl)-3-(3,5-dimethoxy-4-methylphenyl)-3-hydroxypropyl]pyrrol-3-yl]acetic acid
Show/Hide
|
C28H33NO5
|
1
|
1 |
IC50 = 61 nM
|
|
|
CP0477579
|
2-[4-[(2S)-2-[(S)-(3,5-dimethoxy-4-methylphenyl)-hydroxymethyl]-5-phenylpentyl]phenyl]acetic acid
Show/Hide
|
C29H34O5
|
1
|
1 |
IC50 = 61 nM
|
|
|
CP0477605
|
2-[4-[[(3,5-dimethoxy-4-methylbenzoyl)-(3-phenylpropyl)amino]methyl]phenoxy]benzoic acid
Show/Hide
|
C33H33NO6
|
1
|
1 |
IC50 = 71 nM
|
|
|
CP0422336
|
2-[4-[[(3,5-dimethoxybenzoyl)-(3-phenylpropyl)amino]methyl]phenoxy]benzoic acid
Show/Hide
|
C32H31NO6
|
1
|
1 |
IC50 = 89 nM
|
|
|
CP0248077
|
2-[4-[[(3,5-dimethoxy-4-methylbenzoyl)-(3-phenylpropyl)amino]methyl]phenoxy]acetic acid
Show/Hide
|
C28H31NO6
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0551370
|
2-[4-[[(3,5-dimethoxy-4-methylbenzoyl)-(3-phenylpropyl)amino]methyl]phenoxy]-6-methylbenzoic acid
Show/Hide
|
C34H35NO6
|
1
|
1 |
IC50 = 100 nM
|
|
|
CP0567434
|
1-[(2S)-2-[(S)-(3,5-dimethoxy-4-methylphenyl)-hydroxymethyl]-5-phenylpentyl]pyrrole-3-carboxylic acid
Show/Hide
|
C26H31NO5
|
1
|
1 |
IC50 = 120 nM
|
|
|
CP0465057
|
2-[4-[[3-phenylpropyl-(3,4,5-trimethoxybenzoyl)amino]methyl]phenoxy]benzoic acid
Show/Hide
|
C33H33NO7
|
1
|
1 |
IC50 = 130 nM
|
|
|
CP0481815
|
3-[4-[[(3,5-dimethoxybenzoyl)-(3-phenylpropyl)amino]methyl]phenoxy]benzoic acid
Show/Hide
|
C32H31NO6
|
1
|
1 |
IC50 = 140 nM
|
|
|
CP0569670
|
2-[4-[[(3,5-dimethoxy-4-methylbenzoyl)-(3-phenylpropyl)amino]methyl]phenoxy]-3-methylbenzoic acid
Show/Hide
|
C34H35NO6
|
1
|
1 |
IC50 = 140 nM
|
|
|
CP0248075
|
2-[4-[[(3,5-dimethoxy-4-methylbenzoyl)-(3-phenylpropyl)amino]methyl]phenyl]acetic acid
Show/Hide
|
C28H31NO5
|
1
|
1 |
IC50 = 160 nM
|
|
|
CP0511839
|
2-[1-[(2S)-2-[(S)-(3,5-dimethoxy-4-methylphenyl)-hydroxymethyl]-5-phenylpentyl]imidazol-4-yl]acetic acid
Show/Hide
|
C26H32N2O5
|
1
|
1 |
IC50 = 180 nM
|
|
|
CP0507011
|
2-[4-[[(3,5-dimethoxy-4-methylbenzoyl)-[3-(3-fluorophenyl)propyl]amino]methyl]phenyl]acetic acid
Show/Hide
|
C28H30FNO5
|
1
|
1 |
IC50 = 190 nM
|
|
|
CP0445697
|
2-[2-[4-[[(3,5-dimethoxybenzoyl)-(3-phenylpropyl)amino]methyl]phenyl]phenyl]acetic acid
Show/Hide
|
C33H33NO5
|
1
|
1 |
IC50 = 210 nM
|
|
|
CP0530977
|
2-[4-[[(3,5-dimethoxy-4-methylbenzoyl)-[3-(2-fluorophenyl)propyl]amino]methyl]phenyl]acetic acid
Show/Hide
|
C28H30FNO5
|
1
|
1 |
IC50 = 220 nM
|
|
|
CP0575347
|
(1S,3S)-3-[4-[4-[[(4-chlorophenyl)methoxycarbonylamino]methyl]-3-methyl-1,2-oxazol-5-yl]phenoxy]cyclohexane-1-carboxylic acid
Show/Hide
|
C26H27ClN2O6
|
1
|
1 |
IC50 = 227 nM
|
|
|
CP0511815
|
3-[2-[4-[[(3,5-dimethoxybenzoyl)-(3-phenylpropyl)amino]methyl]phenyl]phenyl]propanoic acid
Show/Hide
|
C34H35NO5
|
1
|
1 |
IC50 = 230 nM
|
|
|
CP0477628
|
2-[4-[[(3,5-dimethoxybenzoyl)-(3-phenylpropyl)amino]methyl]phenyl]benzoic acid
Show/Hide
|
C32H31NO5
|
1
|
1 |
IC50 = 260 nM
|
|
|
CP0530873
|
2-[4-[[(3,5-dimethylbenzoyl)-(3-phenylpropyl)amino]methyl]phenyl]benzoic acid
Show/Hide
|
C32H31NO3
|
1
|
1 |
IC50 = 260 nM
|
|
|
CP0450341
|
2-[4-[[3-phenylpropyl-(3,4,5-trimethoxybenzoyl)amino]methyl]phenyl]benzoic acid
Show/Hide
|
C33H33NO6
|
1
|
1 |
IC50 = 390 nM
|
|
|
CP0511840
|
2-[4-[2-(3,5-dimethoxy-4-methylbenzoyl)-5-phenylpentyl]phenyl]acetic acid
Show/Hide
|
C29H32O5
|
1
|
1 |
IC50 = 460 nM
|
|
|
CP0489959
|
2-[1-[(2S)-2-[(S)-(3,5-dimethoxy-4-methylphenyl)-hydroxymethyl]-5-phenylpentyl]-3,5-dimethylpyrazol-4-yl]acetic acid
Show/Hide
|
C28H36N2O5
|
1
|
1 |
IC50 = 520 nM
|
|
|
CP0558532
|
(1S,3S)-3-[6-[4-[(benzylsulfonylamino)methyl]-3-methyl-1,2-oxazol-5-yl]-2-methylpyridin-3-yl]oxycyclohexane-1-carboxylic acid
Show/Hide
|
C25H29N3O6S
|
1
|
1 |
IC50 = 620 nM
|
|
|
CP0555797
|
3-[3-[(3,5-dimethoxy-4-methylbenzoyl)-(3-phenylpropyl)amino]propoxy]benzoic acid
Show/Hide
|
C29H33NO6
|
1
|
1 |
IC50 = 680 nM
|
|
|
CP0567605
|
2-[4-[[(3-methoxybenzoyl)-(3-phenylpropyl)amino]methyl]phenyl]benzoic acid
Show/Hide
|
C31H29NO4
|
1
|
1 |
IC50 = 1300 nM
|
|
|
CP0530978
|
2-[4-[[(3-methylbenzoyl)-(3-phenylpropyl)amino]methyl]phenyl]benzoic acid
Show/Hide
|
C31H29NO3
|
1
|
1 |
IC50 = 1700 nM
|
|
|
CP0465056
|
2-[4-[[(2-methoxybenzoyl)-(3-phenylpropyl)amino]methyl]phenyl]benzoic acid
Show/Hide
|
C31H29NO4
|
1
|
1 |
IC50 = 3300 nM
|
|
|
CP0445696
|
2-[4-[[(3,4-dimethoxybenzoyl)-(3-phenylpropyl)amino]methyl]phenyl]benzoic acid
Show/Hide
|
C32H31NO5
|
1
|
1 |
IC50 = 3700 nM
|
|
|
CP0511814
|
2-[4-[[(4-methoxybenzoyl)-(3-phenylpropyl)amino]methyl]phenyl]benzoic acid
Show/Hide
|
C31H29NO4
|
1
|
1 |
IC50 = 4400 nM
|
|
|
CP0566615
|
2-[4-[[(3-fluorobenzoyl)-(3-phenylpropyl)amino]methyl]phenyl]benzoic acid
Show/Hide
|
C30H26FNO3
|
1
|
1 |
IC50 = 5500 nM
|
|
|
CP0455953
|
2-[4-[[(3,5-dimethoxy-4-methylbenzoyl)-(4-phenylbutyl)amino]methyl]phenoxy]acetic acid
Show/Hide
|
C29H33NO6
|
1
|
1 |
IC50 = 6600 nM
|
|
|
CP0567604
|
2-[4-[[(3,5-dimethoxy-4-methylbenzoyl)-(2-phenylethyl)amino]methyl]phenoxy]acetic acid
Show/Hide
|
C27H29NO6
|
1
|
1 |
IC50 > 10000 nM
|
|
|
CP0445695
|
2-[4-[[benzoyl(3-phenylpropyl)amino]methyl]phenyl]benzoic acid
Show/Hide
|
C30H27NO3
|
1
|
1 |
IC50 = 12100 nM
|
|
|
CP0387271
|
4-(2-ethylbutyl)-N-[3-(4-fluorophenoxy)-5-pyridin-4-yloxyphenyl]-4-hydroxypiperidine-1-carboxamide
Show/Hide
|
C29H34FN3O4
|
1
|
1 |
IC50 > 25000 nM
|
|
|
CP0398647
|
N-[3,5-bis(4-fluorophenoxy)phenyl]-4-(2-ethylbutyl)-4-hydroxypiperidine-1-carboxamide
Show/Hide
|
C30H34F2N2O4
|
1
|
1 |
IC50 > 25000 nM
|
|
|
CP0398735
|
N-[3-(4-cyanophenoxy)-5-(4-fluorophenoxy)phenyl]-4-(2-ethylbutyl)-4-hydroxypiperidine-1-carboxamide
Show/Hide
|
C31H34FN3O4
|
1
|
1 |
IC50 > 25000 nM
|
|
|
CP0411434
|
4-(2-ethylbutyl)-N-[3-(4-fluorophenoxy)-5-pyridin-2-yloxyphenyl]-4-hydroxypiperidine-1-carboxamide
Show/Hide
|
C29H34FN3O4
|
1
|
1 |
IC50 > 25000 nM
|
|
|
CP0477277
|
4-(2-ethylbutyl)-N-[3-(4-fluorophenoxy)-5-pyridin-3-yloxyphenyl]-4-hydroxypiperidine-1-carboxamide
Show/Hide
|
C29H34FN3O4
|
1
|
1 |
IC50 > 25000 nM
|
|
|
CP0355224
|
4-(2-ethylbutyl)-N-[3-(4-fluorophenoxy)-5-[4-(methylcarbamoyl)phenoxy]phenyl]-4-hydroxypiperidine-1-carboxamide
Show/Hide
|
C32H38FN3O5
|
1
|
1 |
IC50 > 800 nM
|
|
|
CP0375037
|
N-[3-(4-carbamoylphenoxy)-5-(4-fluorophenoxy)phenyl]-4-(2-ethylbutyl)-4-hydroxypiperidine-1-carboxamide
Show/Hide
|
C31H36FN3O5
|
1
|
1 |
IC50 > 800 nM
|
|
|
CP0379497
|
4-(2-ethylbutyl)-N-[3-(4-fluorophenoxy)-5-(4-sulfamoylphenoxy)phenyl]-4-hydroxypiperidine-1-carboxamide
Show/Hide
|
C30H36FN3O6S
|
1
|
1 |
IC50 > 800 nM
|
|
|
CP0387270
|
N-[3-(3-carbamoylphenoxy)-5-(4-fluorophenoxy)phenyl]-4-(2-ethylbutyl)-4-hydroxypiperidine-1-carboxamide
Show/Hide
|
C31H36FN3O5
|
1
|
1 |
IC50 > 800 nM
|
|
|
CP0388589
|
N-[3-[4-(dimethylcarbamoyl)phenoxy]-5-(4-fluorophenoxy)phenyl]-4-(2-ethylbutyl)-4-hydroxypiperidine-1-carboxamide
Show/Hide
|
C33H40FN3O5
|
1
|
1 |
IC50 > 800 nM
|
|
|
CP0398734
|
N-[3-(2-carbamoylphenoxy)-5-(4-fluorophenoxy)phenyl]-4-(2-ethylbutyl)-4-hydroxypiperidine-1-carboxamide
Show/Hide
|
C31H36FN3O5
|
1
|
1 |
IC50 > 800 nM
|
|
|
CP0411436
|
4-(2-ethylbutyl)-N-[3-(4-fluorophenoxy)-5-(4-methylsulfonylphenoxy)phenyl]-4-hydroxypiperidine-1-carboxamide
Show/Hide
|
C31H37FN2O6S
|
1
|
1 |
IC50 > 800 nM
|
|
|
CP0445815
|
2-[4-[[(3,5-dimethoxy-4-methylbenzoyl)-[3-(4-fluorophenyl)propyl]amino]methyl]phenyl]acetic acid
Show/Hide
|
C28H30FNO5
|
1
|
1 |
IC50 > 1000 nM
|
|
|
CP0477580
|
2-[4-[[(3,5-dimethoxy-4-methylbenzoyl)-[(E)-3-phenylprop-2-enyl]amino]methyl]phenyl]acetic acid
Show/Hide
|
C28H29NO5
|
1
|
1 |
IC50 > 1000 nM
|
|
|
CP0567606
|
4-[[(3,5-dimethoxy-4-methylbenzoyl)-(3-phenylpropyl)amino]methyl]benzoic acid
Show/Hide
|
C27H29NO5
|
1
|
1 |
IC50 > 1000 nM
|
|
|
CP0905898
|
3-[1-[(2S,3S)-3-(3,5-dimethoxy-4-methyl-phenyl)-3-hydroxy-2-(indan-2-ylmethyl)propyl]pyrrol-3-yl]-2,3-ditritio-propanoic acid
Show/Hide
|
C29H35NO5
|
6
|
1 |
Kd = 0.34 nM
|
|
|
2 |
Kd = 0.49 nM
|
|
|
3 |
Kd = 0.74 nM
|
|
|
4 |
Kd = 1.26 nM
|
|
|
5 |
Kd = 2.34 nM
|
|
|
6 |
Kd = 22.5 nM
|
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CP0867590
|
2-[4-[[(3,5-dimethoxy-4-methyl-benzoyl)-(3-phenyl-2,3-ditritio-propyl)amino]methyl]phenyl]acetic acid
Show/Hide
|
C28H31NO5
|
4
|
1 |
Kd = 5.96 nM
|
|
|
2 |
Kd = 6.54 nM
|
|
|
3 |
Kd = 8.12 nM
|
|
|
4 |
Kd = 10.2 nM
|
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|