US9688710, 116 4-(4-(2-methyl-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran-2-yl)benzyl)phenyl)-N-(1-(4-methylpiperazine-1-carbonyl)cyclopropyl)butanamide

US9688710, 120 N-(2-methyl-1-(4-methylpiperidin-1-yl)-1-oxopropan-2-yl)-4-(4-(2-methyl-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran-2-yl)benzyl)phenyl)butanamide

US9688710, 132 N-(1-((2-(dimethylamino)ethyl)(methyl)amino)-2-methyl-1-oxopropan-2-yl)-4-(4-(2-methyl-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran-2-yl)benzyl)phenyl)butanamide

US9688710, 113 N-(2-methyl-1-(4-methylpiperazin-1-yl)-1-oxopropan-2-yl)-4-(4-(2-methyl-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylsulfinyl)tetrahydro-2H-pyran-2-yl)benzyl)phenyl)butanamide

US9688710, 146 (3R,4R,5S,6R)-2-(3-(4-(3-((3-(dimethylamino)-2,2-dimethylpropyl)amino)propoxy)benzyl)-4-methylphenyl)-6-(methylthio)tetrahydro-2H-pyran-3,4,5-triol

US9688710, 136 N-(1-((2-(dimethylamino)ethyl)amino)-2-methyl-1-oxopropan-2-yl)-4-(4-(2-methyl-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran-2-yl)benzyl)phenyl)butanamide

US9688710, 104 2,2-dimethyl-3-((4-(4-(2-methyl-5-((3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran-2-yl)benzyl)phenyl)butyl)amino)propanamide

4-[4-[[2-chloro-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-methylsulfanyloxan-2-yl]phenyl]methyl]phenoxy]-N-(1-hydroxy-2-methylpropan-2-yl)butanamide

US9688710, 147 N-(2-methyl-1-((1-methylpiperidin-4-yl)amino)-1-oxopropan-2-yl)-4-(4-(2-methyl-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran-2-yl)benzyl)phenyl)butanamide

US9688710, 45 N-(2-methyl-1-(4-methylpiperazin-1-yl)-1-oxopropan-2-yl)-4-(4-(2-methyl-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran-2-yl)benzyl)phenoxy)butanamide

US9688710, 135 (3R,4R,5S,6R)-2-(3-(4-(3-((1-hydroxy-2-methylpropan-2-yl)amino)propoxy)benzyl)-4-methylphenyl)-6-(methylthio)tetrahydro-2H-pyran-3,4,5-triol

US9688710, 127 N-(2,2-dimethyl-3-(4-methylpiperazin-1-yl)-3-oxopropyl)-4-(4-(2-methyl-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran-2-yl)benzyl)phenyl)butanamide

US9688710, 124 4-(4-(2-methyl-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran-2-yl)benzyl)phenyl)-N-(2-(4-methylpiperazin-1-yl)-2-oxoethyl)butanamide

US9688710, 129 2-methyl-2-((4-(4-(2-methyl-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran-2-yl)benzyl)phenyl)butyl)amino)-1-(4-methylpiperazin-1-yl)propan-1-one

US9688710, 4 4-(4-(2-methyl-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran-2-yl)benzyl)phenyl)butanoicacid

US9688710, 37 2-methyl-2-(2-(4-(2-methyl-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran-2-yl)benzyl)phenoxy)acetamido)propanamide

LP-802034

US9688710, 149 1-(1-hydroxy-2-methylpropan-2-yl)-3-(2-(4-(2-methyl-5-((3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran-2-yl)benzyl)phenoxy)ethyl)urea

(2S,3R,4R,5S,6R)-2-[7-[(4-ethylphenyl)methyl]-2,3-dihydro-1H-inden-5-yl]-6-(hydroxymethyl)oxane-3,4,5-triol

1-(2,4-dihydroxy-6-{[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy}phenyl)-3-(4-hydroxyphenyl)propan-1-one

US8614195, 4

US8614195, 2e

US8614195, 2c

ethyl 1-(4-nitrophenyl)-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate

US9688710, 2 4-(4-(2-chloro-5-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(methylthio)tetrahydro-2H-pyran-2-yl)benzyl)phenoxy)butanoic acid

ethyl 1-(2-nitrophenyl)-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate

US8614195, 2a

ethyl 1-phenyl-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate

ethyl 1-(2-bromophenyl)-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate

US8614195, 2b

ethyl 1-(3-nitrophenyl)-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate

ethyl 1-dibenzofuran-3-yl-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate

ethyl 1-[4-(trifluoromethoxy)phenyl]-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate

ethyl 1-(4-fluorophenyl)-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate

ethyl 1-(4-methylphenyl)-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate

ethyl 1-(4-phenylphenyl)-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate

ethyl 1-(2,4-dichlorophenyl)-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate

(2S,3R,4R,5S,6R)-2-[4-chloro-3-[(4-cyclopropylphenyl)methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol

ethyl 1-[2-(trifluoromethyl)phenyl]-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate

ethyl 1-(2-methoxydibenzofuran-3-yl)-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate

ethyl 1-(4-bromophenyl)-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate

(2S,3R,4R,5S,6R)-2-[4-chloro-3-[(4-ethenylphenyl)methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol

ethyl 1-(2,5-dimethoxyphenyl)-5-[(1S,2S,3S)-1,2,3-trihydroxybutyl]triazole-4-carboxylate

(2S,3R,4R,5S,6R)-2-{4-chloro-3-[(4-ethoxyphenyl)methyl]phenyl}-6-(hydroxymethyl)oxane-3,4,5-triol

US8614195, 3

(2S,3R,4R,5S,6R)-2-(4-chloro-3-(4-hydroxybenzyl)phenyl)-6-(hydroxymethyl)tetrahydro-2H-pyran-3,4,5-triol

US8614195, 2g

(2S,3R,4R,5S,6R)-2-[4-chloro-3-[(4-ethynylphenyl)methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol

(2S,3R,4R,5S,6R)-2-[4-chloro-3-[[4-(1-hydroxycyclopropyl)phenyl]methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol

US8614195, 2f

(2S,3R,4R,5S,6R)-2-[4-chloro-3-[[4-(2-prop-2-enoxyethoxy)phenyl]methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol

(2S,3R,4R,5S,6R)-2-[4-chloro-3-[[4-(2-cyclopropyloxyethoxy)phenyl]methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol

US8614195, 3a

(2S,3R,4R,5S,6R)-2-[4-chloro-3-[[4-(2-prop-2-ynoxyethoxy)phenyl]methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol

(2S,3R,4R,5S,6R)-2-[4-chloro-3-[[4-(2-cyclopentyloxyethoxy)phenyl]methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol

3-phenyl-1-(2,4,6-trihydroxyphenyl)-1-propanone

2-[4-[[2-chloro-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]phenoxy]acetic acid

3-(4-fluorophenyl)-1-(2,4,6-trihydroxyphenyl)propan-1-one

3-(4-fluorophenyl)-1-[2,4,6-trihydroxy-3-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]propan-1-one

3-(4-methylphenyl)-1-(2,4,6-trihydroxyphenyl)propan-1-one

3-phenyl-1-[2,4,6-trihydroxy-3-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]propan-1-one

(2S,3R,4R,5S,6R)-2-[4-chloro-3-[[4-(3-cyclopropylprop-2-ynoxy)phenyl]methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol

(2S,3R,4R,5S,6R)-2-[4-chloro-3-[[4-[2-(1-methylcyclopropyl)oxyethoxy]phenyl]methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol

ethyl 2-[4-[[2-chloro-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]phenoxy]acetate

(2S,3R,4R,5S,6R)-2-[4-chloro-3-[[4-(2-cyclopropyloxyethyl)phenyl]methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol

(2S,3R,4R,5S,6R)-2-[4-chloro-3-[[4-[1-(methoxymethyl)cyclopropyl]phenyl]methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol

N-[[4-[[2-chloro-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]phenyl]methyl]-N-cyclopropylacetamide

(2S,3R,4R,5S,6R)-2-[4-chloro-3-[[4-(cyclopropyloxymethyl)phenyl]methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol

(2S,3R,4R,5S,6R)-2-[4-chloro-3-[[4-(2-cyclohexyloxyethoxy)phenyl]methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol

4-[[2-chloro-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]benzonitrile

(2S,3R,4R,5S,6R)-2-[4-chloro-3-[[4-(2-hydroxyethoxy)phenyl]methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol

(E)-3-(4-methylphenyl)-1-(2,4,6-trihydroxyphenyl)prop-2-en-1-one

3-(4-methylphenyl)-1-[2,4,6-trihydroxy-3-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]propan-1-one

3-(4-propoxyphenyl)-1-(2,4,6-trihydroxyphenyl)propan-1-one

3-(4-hydroxyphenyl)-1-(2,4,6-trihydroxyphenyl)propan-1-one

3-(4-methoxyphenyl)-1-(2,4,6-trihydroxyphenyl)propan-1-one

3-(4-methoxyphenyl)-1-[2,4,6-trihydroxy-3-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]propan-1-one

3-(4-ethoxyphenyl)-1-[2,4,6-trihydroxy-3-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]propan-1-one

3-(4-ethoxyphenyl)-1-(2,4,6-trihydroxyphenyl)propan-1-one

3-(4-propoxyphenyl)-1-[2,4,6-trihydroxy-3-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]propan-1-one

3-(4-hydroxyphenyl)-1-[2,4,6-trihydroxy-3-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]propan-1-one

(E)-3-Phenyl-1-(2,4,6-trihydroxy-phenyl)-propenone

4-FLUORO-2',4',6'-TRIHYDROXYCHALCONE

(E)-3-(4-prop-2-enoxyphenyl)-1-(2,4,6-trihydroxyphenyl)prop-2-en-1-one

(E)-3-(4-ethoxyphenyl)-1-(2,4,6-trihydroxyphenyl)prop-2-en-1-one

4-BROMO-2',4',6'-TRIHYDROXYCHALCONE

(2S,3R,4R,5S,6R)-2-[4-chloro-3-[[4-(2-cyclobutyloxyethoxy)phenyl]methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol

4-METHOXYL-2',4',6'-TRIHYDROXYCHALCONE

(E)-3-(4-phenylmethoxyphenyl)-1-(2,4,6-trihydroxyphenyl)prop-2-en-1-one

(2S,3R,4R,5S,6R)-2-[4-chloro-3-[(4-methoxynaphthalen-1-yl)methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol

(2S,3R,4R,5S,6R)-2-[4-chloro-3-[[4-[2-[(3R)-oxolan-3-yl]oxyethoxy]phenyl]methyl]phenyl]-6-(hydroxymethyl)oxane-3,4,5-triol

4-[[2-chloro-5-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]phenyl]methyl]benzamide

(2S,3R,4R,5S,6R)-2-[3-[[4-(2-but-2-ynoxyethoxy)phenyl]methyl]-4-chlorophenyl]-6-(hydroxymethyl)oxane-3,4,5-triol

(2S,3R,4R,5S,6R)-2-[3-[(4-but-2-ynoxyphenyl)methyl]-4-chlorophenyl]-6-(hydroxymethyl)oxane-3,4,5-triol