Brief Information of the Cell Line and Protein
Cell Line ID: CL000011 , CHO
Synonyms
Chinese Hamster Ovary
CHO-ori
Category Spontaneously immortalized cell line
Organism
Cricetulus griseus (Chinese hamster)
Cellosaurus ID
CVCL_0213
Protein ID: PT03188 , Vasopressin V1b receptor
Gene Name AVPR1B
Organism Rattus norvegicus, Rat
Protein Classification Membrane receptor
Uniprot ID P48974
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000011  Protein ID: PT03188
 
Compound ID Compound Name Compound Formula
CP0140566
2-[2-(3-methoxyphenyl)-4-oxo-6-(3-piperidin-1-ylpropoxy)quinazolin-3-yl]-N-propan-2-ylacetamide
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C28H36N4O4
 1
1
IC50 = 2 nM
   TI
   LI
   LO
   TS
CP0103104
2-(2-(3-chlorophenyl)-4-oxo-6-(3-(piperidin-1-yl)propoxy)quinazolin-3(4H)-yl)-N-isopropylacetamide
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C27H33ClN4O3
 1
1
IC50 = 4 nM
   TI
   LI
   LO
   TS
CP0195952
(2S,4R)-1-((R)-5-chloro-1-(2,4-dimethoxyphenylsulfonyl)-3-(2-methoxyphenyl)-2-oxoindolin-3-yl)-4-hydroxy-N,N-dimethylpyrrolidine-2-carboxamide
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C30H32ClN3O8S
 1
1
Ki = 1 nM
   TI
   LI
   LO
   TS
CP0852136
(R)-4-chloro-3-(5-chloro-1-(2,4-dimethoxybenzyl)-3-methyl-2-oxoindolin-3-yl)-N-ethyl-N-(pyridin-3-ylmethyl)benzamide hydrochloride
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C33H32Cl3N3O4
 1
1
Ki = 46 nM
   TI
   LI
   LO
   TS