| Compound ID |
Compound Name |
Compound Formula |
|
CP0398972
|
Aib-Val-Aib-Glu-lle-Gln-Leu-Nle-His-Gln-Arg-Ala-Lys-Tyr
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|
C76H127N23O19
|
3
|
| 1 |
IC50 = 6.87 nM
|
|
|
| 2 |
IC50 = 55.4 nM
|
|
|
| 3 |
Kd = 21.6 nM
|
|
|
|
CP0398970
|
Aib-Val-Aib-Glu-lle-Gln-Leu-Nle-His-Gln-Har-Ala-Lys-Tyr
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|
C77H129N23O19
|
1
|
| 1 |
IC50 = 7.2 nM
|
|
|
|
CP0423355
|
Aib-Val-Aib-Glu-lle-Gln-Leu-Nle-His-Gln-Arg-Ala-Fly-Tyr
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|
C96H137N23O23
|
1
|
| 1 |
IC50 = 13.5 nM
|
|
|
|
CP0423356
|
Aib-Val-Aib-Glu-lle-Gln-Leu-Nle-His-Gln-Arg-Ala-Lys-Tyr-Fly
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|
C102H149N25O24
|
1
|
| 1 |
IC50 = 98.2 nM
|
|
|
|
CP0053165
|
(3S,5S)-5-[(E)-2-cyclopropylethenyl]-3-ethyl-6,7-difluoro-5-(trifluoromethyl)-1H-4,1-benzoxazepin-2-one
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|
C17H16F5NO2
|
3
|
| 1 |
IC50 = 990 nM
|
|
|
| 2 |
IC50 = 5780 nM
|
|
|
| 3 |
IC50 = 68000 nM
|
|
|
|
CP0431771
|
Ala-Val-Ala-Glu-lle-Gln-Leu-Nle-His-Gln-Har-Ala-Lys-Trp-Tyr
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|
C86H135N25O20
|
1
|
| 1 |
IC50 = 2187 nM
|
|
|
|
CP0423354
|
Ala-Val-Ala-Glu-lle-Gln-Leu-Met-His-Gln-Har-Ala-Lys-Trp-Fly
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|
C102H146N26O23S
|
1
|
| 1 |
IC50 = 10130 nM
|
|
|
|
CP0436332
|
Ala-Val-Ala-Glu-lle-Gln-Leu-Met-His-Gln-Har-Ala-Lys-Trp
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|
C76H124N24O18S
|
1
|
| 1 |
IC50 = 10484 nM
|
|
|
|
CP0431898
|
Ala-Val-Ala-Glu-lle-Gln-Leu-Nle-His-Gln-Har-Ala-Lys-Tyr
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|
C75H125N23O19
|
1
|
| 1 |
IC50 = 10560 nM
|
|
|