Brief Information of the Cell Line and Protein
Cell Line ID: CL000787 , HKRK-B28
Category Spontaneously immortalized cell line
Organism
Sus scrofa (Pig)
Cellosaurus ID
CVCL_0391
Protein ID: PT02986 , Parathyroid hormone/parathyroid hormone-related peptide receptor
Gene Name PTH1R
Organism Homo sapiens, Human
Protein Classification Membrane receptor
Uniprot ID Q03431
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000787  Protein ID: PT02986
 
Compound ID Compound Name Compound Formula
CP0398972
Aib-Val-Aib-Glu-lle-Gln-Leu-Nle-His-Gln-Arg-Ala-Lys-Tyr
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C76H127N23O19
 3
1
IC50 = 6.87 nM
   TI
   LI
   LO
   TS
2
IC50 = 55.4 nM
   TI
   LI
   LO
   TS
3
Kd = 21.6 nM
   TI
   LI
   LO
   TS
CP0398970
Aib-Val-Aib-Glu-lle-Gln-Leu-Nle-His-Gln-Har-Ala-Lys-Tyr
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C77H129N23O19
 1
1
IC50 = 7.2 nM
   TI
   LI
   LO
   TS
CP0423355
Aib-Val-Aib-Glu-lle-Gln-Leu-Nle-His-Gln-Arg-Ala-Fly-Tyr
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C96H137N23O23
 1
1
IC50 = 13.5 nM
   TI
   LI
   LO
   TS
CP0423356
Aib-Val-Aib-Glu-lle-Gln-Leu-Nle-His-Gln-Arg-Ala-Lys-Tyr-Fly
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C102H149N25O24
 1
1
IC50 = 98.2 nM
   TI
   LI
   LO
   TS
CP0053165
(3S,5S)-5-[(E)-2-cyclopropylethenyl]-3-ethyl-6,7-difluoro-5-(trifluoromethyl)-1H-4,1-benzoxazepin-2-one
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C17H16F5NO2
 3
1
IC50 = 990 nM
   TI
   LI
   LO
   TS
2
IC50 = 5780 nM
   TI
   LI
   LO
   TS
3
IC50 = 68000 nM
   TI
   LI
   LO
   TS
CP0431771
Ala-Val-Ala-Glu-lle-Gln-Leu-Nle-His-Gln-Har-Ala-Lys-Trp-Tyr
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C86H135N25O20
 1
1
IC50 = 2187 nM
   TI
   LI
   LO
   TS
CP0423354
Ala-Val-Ala-Glu-lle-Gln-Leu-Met-His-Gln-Har-Ala-Lys-Trp-Fly
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C102H146N26O23S
 1
1
IC50 = 10130 nM
   TI
   LI
   LO
   TS
CP0436332
Ala-Val-Ala-Glu-lle-Gln-Leu-Met-His-Gln-Har-Ala-Lys-Trp
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C76H124N24O18S
 1
1
IC50 = 10484 nM
   TI
   LI
   LO
   TS
CP0431898
Ala-Val-Ala-Glu-lle-Gln-Leu-Nle-His-Gln-Har-Ala-Lys-Tyr
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C75H125N23O19
 1
1
IC50 = 10560 nM
   TI
   LI
   LO
   TS