Brief Information of the Cell Line and Protein
Cell Line ID: CL000174 , Raji
Synonyms
RAJI
P1-Raji
GM04671
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0511
Protein ID: PT02583 , Proteasome subunit beta type-1
Gene Name PSMB1
Organism Homo sapiens, Human
Protein Classification Enzyme
Uniprot ID P20618
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000174  Protein ID: PT02583
 
Compound ID Compound Name Compound Formula
CP0045910
(S)-2-azido-N-((S)-1-((S)-1-((S)-4-methyl-1-((R)-2-methyloxiran-2-yl)-1-oxopentan-2-ylamino)-1-oxo-3-phenylpropan-2-ylamino)-1-oxo-3-phenylpropan-2-yl)-3-phenylpropanamide
   Show/Hide
C36H42N6O5
 2
1
IC50 = 120 nM
   TI
   LI
   LO
   TS
2
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0446489
(2S)-2-[[(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-3-(4-methoxyphenyl)propanoyl]amino]-N-[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]-3-phenylpropanamide
   Show/Hide
C37H44N6O6
 2
1
IC50 = 130 nM
   TI
   LI
   LO
   TS
2
IC50 = 180 nM
   TI
   LI
   LO
   TS
CP0475289
(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-N-[(2S)-1-[[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]-4-phenylbutanamide
   Show/Hide
C37H44N6O5
 2
1
IC50 = 160 nM
   TI
   LI
   LO
   TS
2
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0455723
(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-3-(4-methoxycyclohexyl)-N-[(2S)-1-[[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]propanamide
   Show/Hide
C37H50N6O6
 2
1
IC50 = 890 nM
   TI
   LI
   LO
   TS
2
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0446492
(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-N-[(2S)-1-[[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]-3-(4-phenylcyclohexyl)propanamide
   Show/Hide
C39H46N6O5
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0455722
(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-3-(4-cyclohexylcyclohexyl)-N-[(2S)-1-[[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]propanamide
   Show/Hide
C39H52N6O5
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0475291
(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-3-(4-cyclohexylcyclohexyl)-N-[(2S)-1-[[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]propanamide
   Show/Hide
C39H52N6O5
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0482909
(2S)-N-[(2S)-3-(4-cyclohexylcyclohexyl)-1-[[(2S)-1-[[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]amino]-1-oxopropan-2-yl]-4-methyl-2-[(2-morpholin-4-ylacetyl)amino]pentanamide
   Show/Hide
C42H65N5O7
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0534919
(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-3-(4-methylcyclohexyl)-N-[(2S)-1-[[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]propanamide
   Show/Hide
C37H50N6O5
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0420040
(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-3-(4-cyclohexylcyclohexyl)-N-[(2S)-1-[[(2S)-4-methyl-1-[(2R)-2-methyloxiran-2-yl]-1-oxopentan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]propanamide
   Show/Hide
C42H58N6O5
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0420041
(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-3-(4-cyclohexylcyclohexyl)-N-[(2S)-1-[[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]propanamide
   Show/Hide
C39H52N6O5
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0455719
(2S)-2-[[(2S)-2-azido-3-phenylpropanoyl]amino]-N-[(2S)-1-[[(2S)-1-[(2R)-2-methyloxiran-2-yl]-1-oxopropan-2-yl]amino]-1-oxo-3-phenylpropan-2-yl]-3-(4-phenylcyclohexyl)propanamide
   Show/Hide
C39H46N6O5
 1
1
IC50 > 100000 nM
   TI
   LI
   LO
   TS
CP0868641
N-((R)-1-((S)-1-((S)-3-cyclohexyl-1-((R)-2-methyloxiran-2-yl)-1-oxopropan-2-ylamino)-3-(1H-indol-3-yl)-1-oxopropan-2-ylamino)-1-oxopropan-2-yl)-3-methyl-1H-indene-2-carboxamide
   Show/Hide
C37H44N4O5
 1
1
IC50 > 1000 nM
   TI
   LI
   LO
   TS