Brief Information of the Cell Line and Protein
Cell Line ID: CL000197 , MG-63
Synonyms
M-G63
MG63
Category Cancer cell line
Organism
Homo sapiens (Human)
Cellosaurus ID
CVCL_0426
Protein ID: PT02513 , Steroid hormone receptor ERR1
Gene Name ESRRA
Organism Homo sapiens, Human
Protein Classification Transcription factor
Uniprot ID P11474
Table of Molecular Bioactivities Related to the Cell Line and Protein
Cell Line ID: CL000197  Protein ID: PT02513
 
Compound ID Compound Name Compound Formula
CP0549469
2-tert-butyl-4-(2,3-dimethylbenzimidazol-5-yl)oxyphenol
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C19H22N2O2
 1
1
EC50 = 1100 nM
   TI
   LI
   LO
   TS
CP0469262
5-[[4-[[6-(3-tert-butyl-4-hydroxyphenoxy)-1-methylbenzimidazol-2-yl]methoxy]phenyl]methyl]-1,3-thiazolidine-2,4-dione
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C29H29N3O5S
 1
1
EC50 = 5200 nM
   TI
   LI
   LO
   TS
CP0517157
1-[4-(3-tert-butyl-4-hydroxyphenoxy)phenyl]ethanone
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C18H20O3
 1
1
EC50 = 5400 nM
   TI
   LI
   LO
   TS
CP0549472
1-[4-(3-tert-butyl-4-hydroxyphenoxy)-3-chlorophenyl]ethanone
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C18H19ClO3
 1
1
EC50 = 5900 nM
   TI
   LI
   LO
   TS
CP0444766
2-tert-butyl-4-(3-methyl-2-phenylbenzimidazol-5-yl)oxyphenol
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C24H24N2O2
 1
1
EC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0469234
N-[3-chloro-4-(4-chloronaphthalen-1-yl)oxyphenyl]butanamide
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C20H17Cl2NO2
 1
1
EC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0469235
N-(3-chloro-4-naphthalen-1-yloxyphenyl)acetamide
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C18H14ClNO2
 1
1
EC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0517155
N-[3-chloro-4-(4-chloronaphthalen-1-yl)oxyphenyl]propanamide
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C19H15Cl2NO2
 1
1
EC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0531925
2-tert-butyl-4-[3-methyl-2-(phenoxymethyl)benzimidazol-5-yl]oxyphenol
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C25H26N2O3
 1
1
EC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0549468
N-[4-(4-chloronaphthalen-1-yl)oxyphenyl]acetamide
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C18H14ClNO2
 1
1
EC50 > 10000 nM
   TI
   LI
   LO
   TS
CP0549470
N-[4-(3-tert-butyl-4-hydroxyphenoxy)-3-chlorophenyl]acetamide
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C18H20ClNO3
 1
1
EC50 > 10000 nM
   TI
   LI
   LO
   TS